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血管生成库
TargetMol

Angiogenesis related Compound Library

血管生成是正常生长和发育过程以及伤口愈合和肉芽组织形成过程中的基本事件,然而异常的血管生成将导致各种疾病,例如肿瘤、糖尿病、免疫病、先兆子痫、肢体缺血等。因此,血管生成已成为治疗这些疾病的药物靶点。例如,血管生成与癌症发生密切相关,肿瘤通过分泌各种生长因子(例如VEGF)和蛋白质诱导毛细血管生成进入肿瘤,为癌细胞提供氧气和其他必需的营养物质,并及时运走代谢废物,血管生成也是肿瘤扩散或转移所必需的。因此血管生成抑制剂用于治疗癌症。此外,诱导血管生成,建立新的侧支循环是治疗缺血性心脑血管疾病(冠心病、脑卒中等)的极佳治疗方式。有效新生血管靶分子的筛选为相关疾病研究带来了广阔前景。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L4800
产品编号: L4800
  • 规格
  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 产品描述:
    • 2300个高潜力的抑制或促进血管生成的小分子集合,可用于药物靶点开发、血管生成机理研究的高通量筛选,高内涵筛选;
    • 包含了目前研究较多潜力的血管生成通路以及S1P、VEGFR、PDGF等相关靶点的热门产品;
    • 包含了Sunitinib Malate、Lenalidomide、sorafenib、Erlotinib等研究成熟的上市药物,以及Vatalanib、Orantinib、2-Methoxyestradiol(Panzem)、Celecoxib等临床药物;
    • 是研究血管生成机理以及药物靶向研究的有效工具;
    • 产品经过临床验证和临床实验,具有生物安全保障和一定的生物活性;
    • 结构多样,药效显著,可渗透细胞;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR和HPLC检测技术保证产品高纯度和高质量;
    • 所有化合物现货供应。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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