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抗结直肠癌化合物库
TargetMol

Anti-Colorectal Cancer Compound Library

结直肠癌(Colorectal Cancer,CRC),又称大肠癌,包括结肠癌和直肠癌,是全球范围内致命的恶性肿瘤之一,严重威胁人类健康,近年来其发病率和死亡率均呈上升趋势,并且发病率随着年龄的增加而增加,人口老龄化和不良生活习惯是主要诱因,缺乏运动、肥胖、抽烟也使得患结直肠癌的风险显著增加。结直肠癌的治疗手段包括手术、放疗、化疗和靶向治疗。早期癌症可以通过手术治愈,晚期转移性癌通常选择化疗联合靶向治疗,研究表明,多个信号通路和靶点的失调与结直肠癌有关,如: VEGFR、EGFR、Wnt/β-catenin、p53、TGF-β等 TargetMol 抗结直肠癌化合物库收集了1880 种与结直肠癌相关的化合物,包括已经报道具有结直肠癌治疗作用的化合物,以及靶向结直肠癌相关靶点的化合物,是抗结直肠癌药物研发的良好工具。

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L2194
产品编号: L2194
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 产品描述:
    • 1880种与结直肠癌相关的化合物,可以用于高通量和高内涵筛选;
    • 部分化合物已上市或已进入临床期;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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