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抗乳腺癌化合物库
TargetMol

Anti-Breast Cancer Compound Library

乳腺癌是乳腺恶性肿瘤,是全球女性发病率较高的癌症,约占女性癌症患者的20%,也是100多个国家癌症死亡的主要原因。近年来全球乳腺癌发病率一直呈上升趋势。 乳腺癌根据病理分型可分为非浸润性癌,早期浸润性癌,浸润性癌。根据分子分型可分为雌激素受体阳性乳腺癌(ER+PR+HER2-),HER2阳性乳腺癌(ER-PR-HER2+),三阴性乳腺癌(ER-PR-HER2-)。不同类型的乳腺癌,从治疗方法到预后都是非常不同,需要针对已经明确的致癌位点,探索相关靶点来设计相应的药物。 TargetMol 抗乳腺癌库收集了2440 种与乳腺癌相关的化合物,包含了已经报道的有乳腺癌治疗作用的化合物,以及相关的靶点通路(HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA 等),是乳腺癌药物研发的良好工具。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L2191
产品编号: L2191
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 产品描述:
    • 2440种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
    • 靶点包含HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA等;
    • 部分化合物已上市或已进入临床期;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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