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抗癌临床化合物库
TargetMol

Anti-Cancer Clinical Compound Library

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号(例如治疗药物)诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力,表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

抗癌活性的药物是临床研究的热点之一,根据文献报道和有关公开资料,我们收集了2760 个具有抗癌活性或潜在抗癌活性的处于临床试验阶段的化合物,组成抗癌临床化合物库,可用于癌症相关研究及高通量高内涵筛选。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L2120
产品编号: L2120
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
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技术资料

产品描述
  • 产品描述:
    • 2760个具有抗癌活性小分子的独特集合,可用于高通量高内涵筛选;
    • 生物活性已经临床前实验证实,所有化合物均已进入临床实验阶段的抗癌化合物;
    • 包括肺癌、乳腺癌、白血病、淋巴瘤等15种癌症,是癌症相关研究的有效筛选工具;
    • 作用靶点涉及PI3K,HDAC, mTOR, CDK, JAK 等癌症相关靶点;
    • 结构多样,药效显著,可渗透细胞;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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