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抗纤维化化合物库
TargetMol

Anti-Fibrosis Compound Library

纤维化(fibrosis)是一种病理改变,主要表现为器官组织内纤维结缔组织增多,实质细胞减少,持续进展可致器官结构破坏和功能减退,乃至衰竭,严重威胁人类健康和生命。纤维化可发生于多种器官,常见的包括肺脏、肝脏、肾脏、骨髓等。纤维化通常由各种刺激导致的慢性炎症性反应引起,包括:持续性感染,自身免疫反应,过敏性反应,化学刺激,射线和组织损伤等。

TargetMol 抗纤维化化合物库收集了1800 种抗纤维化分子和潜在的抗纤维化分子,包括相关靶点如TGFβ、TNFα、MMP 的抑制剂、抗氧化剂及抗炎分子等,是研究纤维化机制和开发抗纤维化药物的良好工具。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L9810
产品编号: L9810
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
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技术资料

产品描述
  • 产品特性:
    • 1800种潜在的抗纤维化分子,是研究纤维化的有效工具,可以用于高通量筛选和高内涵筛选;
    • 靶点包括TGFβ、TNFα、MMP、EGFR、NADPH-oxidase等;
    • 部分化合物已经得到FDA批准上市;?
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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