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神经退行性疾病化合物库
TargetMol

Anti-Neurodegenerative Disease Compound Library

神经退行性疾病是机体神经元结构或功能逐渐丧失而引发的一类疾病,包括肌萎缩侧索硬化症(Amyotrophiclateral sclerosis,ALS)、帕金森病(Parkinson’s disease,PD)、阿尔茨海默病(Alzheimer disease,AD)、亨廷顿氏病(Huntington’s disease,HD)以及脊髓性肌萎缩症(spinal muscular atrophy,SMA)等,目前这类疾病病因尚不明确并无有效治愈手段,且严重威胁着患者的生活质量。

TargetMol 基于目前的研究现状,收集了2154 种与神经退行性疾病相关的化合物,这些化合物或者对神经退行性疾病有一定的疗效,或者作用于神经退行性疾病相关的靶点,可以用于神经退行性疾病相关的药物研发和机制研究。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L2620
产品编号: L2620
  • 规格
  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
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技术资料

产品描述
  • 产品描述:
    • 2154种与神经退行性疾病相关的化合物,可用于高通量和高内涵筛选;
    • 靶点包括AchE, NMDA, CGRP, β-secretase, γ-secretase, Dopamine Receptor, Adenosine Receptor, 5-HT receptor等;
    • 部分化合物已经得到FDA批准上市;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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化合物库组成
5-HT Receptor
AChR
Dopamine Receptor
Adrenergic Receptor
Apoptosis
Autophagy
GABA Receptor
iGluR
Endogenous Metabolite
GluR
Cholinesterase (ChE)
Histamine Receptor
Opioid Receptor
Others
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Beta Amyloid
PDE
ROS
Monoamine Oxidase
Antibacterial
COX
NF-κB
MAO
JNK
Serotonin Transporter
Potassium Channel
Reactive Oxygen Species
Parasite
Calcium Channel
PPAR
Gamma-secretase
Caspase
GSK-3
Norepinephrine
Sodium Channel
Adenosine Receptor
Cytochromes P450
TNF
Akt
ERK
Influenza Virus
Nrf2
HIV Protease
PI3K
Interleukin
CDK
CaMK
LRRK2
NO Synthase
p38 MAPK
Ferroptosis
Mitophagy
Beta-Secretase
Antifungal
BACE
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Mitochondrial Metabolism
MMP
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Wnt/beta-catenin
DNA/RNA Synthesis
Cannabinoid Receptor
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mTOR
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TRP/TRPV Channel
Src
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IL Receptor
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Bcl-2 Family
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Microtubule Associated
PKC
Trk receptor
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Phospholipase
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Glucosidase
Sirtuin
HDAC
MEK
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glycosidase
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MT Receptor
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MAPK
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Aryl Hydrocarbon Receptor
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AAK1 (AP2 associated kinase 1)
Angiotensin-converting Enzyme (ACE)
Epoxide Hydrolase
PGE Synthase
Antiviral
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Histone Acetyltransferase
transporter
Casein Kinase
c-Fms
IRAK
S6 Kinase
p53
Advanced Glycation End Products
ATPase
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Progesterone Receptor
OCT
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Immunology/Inflammation related
CSF-1R
IAP
Topoisomerase
PAFR
Raf
GRK
Antifection
Monoamine Transporter
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PDGFR
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OXPHOS
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STING
Free radical scavengers
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RSV
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Hydroxylase
FOXO
CGRP Receptor
Gap Junction Protein
FAK
CFTR
FOXO3
Thyroid hormone receptor(THR)
Proteasome
Taste receptor
CAT
NPC1L1
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HCV Protease
Glutaminyl Cyclase
Arrestin
Na+/Ca2+ Exchanger
Reductase
Lipase
Glutathione Peroxidase
GTPase
c-Myc
CaSR
Hck
Serine Protease
Neurotensin Receptor
Glutaminase
ROCK
NR4A
RANKL/RANK
LDLR
IDO
Prolyl Endopeptidase (PREP)
Annexin A
E1/E2/E3 Enzyme
RIP kinase
Adiponectin Receptor
LDL
Hexokinase
HCN Channel
Neuropeptide Y Receptor
Bombesin Receptor
DNA Alkylation
PAK
Somatostatin
Chk
PAD
Cadherin
Orphan receptor
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
Telomerase
SGLT
ATP Citrate Lyase
Lipid
PSMA
MNK
Survivin
OAT
GluCls
PAI-1
Pyroptosis
ALK
Neprilysin
GST
Carboxypeptidase
FKBP
Aromatase
PDK
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Adenosine Deaminase
Cuproptosis
SGK
REV-ERB
Syk
DNA Methyltransferase
Thrombin
Liposome
ROS Kinase
MLK
Vitamin
BTK
NMU2R
NMUR

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