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神经退行性疾病化合物库
TargetMol

Anti-Neurodegenerative Disease Compound Library

神经退行性疾病是机体神经元结构或功能逐渐丧失而引发的一类疾病,包括肌萎缩侧索硬化症(Amyotrophiclateral sclerosis,ALS)、帕金森病(Parkinson’s disease,PD)、阿尔茨海默病(Alzheimer disease,AD)、亨廷顿氏病(Huntington’s disease,HD)以及脊髓性肌萎缩症(spinal muscular atrophy,SMA)等,目前这类疾病病因尚不明确并无有效治愈手段,且严重威胁着患者的生活质量。

TargetMol 基于目前的研究现状,收集了2154 种与神经退行性疾病相关的化合物,这些化合物或者对神经退行性疾病有一定的疗效,或者作用于神经退行性疾病相关的靶点,可以用于神经退行性疾病相关的药物研发和机制研究。

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L2620
产品编号: L2620
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 产品描述:
    • 2154种与神经退行性疾病相关的化合物,可用于高通量和高内涵筛选;
    • 靶点包括AchE, NMDA, CGRP, β-secretase, γ-secretase, Dopamine Receptor, Adenosine Receptor, 5-HT receptor等;
    • 部分化合物已经得到FDA批准上市;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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