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铁死亡化合物库
TargetMol

Ferroptosis Compound Library

铁死亡(ferroptosis)是近年来发现的一种由铁依赖的氧化损伤引起的细胞死亡模式,与凋亡、坏死、自噬不同,铁死亡的特征主要是细胞体积缩小和线粒体膜密度增加,没有典型的细胞凋亡和坏死表现。ferroptosis 与神经系统疾病、肿瘤(特别是乳腺癌、弥漫性大 B 细胞淋巴瘤)、缺血再灌注损伤、肾损伤、动脉粥样硬化、糖尿病、心脏病等疾病有关,进一步深入研究铁死亡的作用机理,研究其在不同疾病类型中的作用,对寻找相关疾病的治疗靶点、靶向药物的研发具有重要意义。

TargetMol 铁死亡化合物库,收集了 950 种与铁死亡通路相关的化合物,靶点包括 GPX4、ROS、p53、Nrf2等,另外还包含了铁螯合剂、抗氧化剂等多种类型小分子,助力您铁死亡通路相关的靶点鉴定和药物研发。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L8700
产品编号: L8700
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
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技术资料

产品描述
  • 产品描述:
    • 950种与铁死亡通路相关的化合物,可用于高通量和高内涵筛选;
    • 靶点含GPX4,ROS,p53,Nrf2等;
    • 部分化合物已被FDA批准上市;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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化合物库组成
ROS
Apoptosis
Reactive Oxygen Species
Autophagy
Ferroptosis
Endogenous Metabolite
Nrf2
PPAR
NF-κB
Lipoxygenase
Antibacterial
Others
Ras
p38 MAPK
COX
p53
MDM-2/p53
Antioxidant
Akt
Antifungal
DNA/RNA Synthesis
Dehydrogenase
Caspase
Parasite
HMG-CoA Reductase
FXR
ERK
Cytochromes P450
Interleukin
JNK
TNF
Bcl-2 Family
Antibiotic
Influenza Virus
HIV Protease
PI3K
NADPH
Glutathione Peroxidase
Raf
Mdm2
HIF/HIF Prolyl-Hydroxylase
NO Synthase
Mitophagy
AMPK
PARP
Calcium Channel
Mitochondrial Metabolism
MMP
VEGFR
CDK
TLR
STAT
NOD-like Receptor (NLR)
Virus Protease
Wnt/beta-catenin
Potassium Channel
TRP/TRPV Channel
Topoisomerase
SARS-CoV
NADPH-oxidase
Proteasome
Rho
GPX
5-HT Receptor
Phosphatase
E1/E2/E3 Enzyme
IL Receptor
Cholinesterase (ChE)
TGF-beta/Smad
P-gp
Estrogen/progestogen Receptor
GSK-3
mTOR
Beta Amyloid
GABA Receptor
AChR
Microtubule Associated
Kras
PKC
EGFR
HSP
Sirtuin
Pyroptosis
HIF
Tyrosinase
ATPase
Src
Reductase
Estrogen Receptor/ERR
HBV
Leukotriene Receptor
MAO
Immunology/Inflammation related
Opioid Receptor
DPP-4
JAK
HSV
IGF-1R
MAPK
Prostaglandin Receptor
GPCR19
IκB/IKK
Anti-infection
Monoamine Oxidase
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HCV Protease
PERK
Histamine Receptor
Photosensitizer
IAP
iGluR
Drug Metabolite
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Xanthine Oxidase
DUB
NOS
ROR
Integrin
Amino Acids and Derivatives
MyD88
LTR
RAAS
PKA
Adrenergic Receptor
Aryl Hydrocarbon Receptor
IDO
UGT
PDE
LDL
Gamma-secretase
Glucosidase
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GluR
Epigenetic Reader Domain
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
Lipid
OXPHOS
Antiviral
Histone Acetyltransferase
Reverse Transcriptase
HDAC
Aromatase
Cannabinoid Receptor
FLT
Sodium Channel
NOD
ROS Kinase
Carbonic Anhydrase
Transferase
Ferroportin
DNA Alkylator/Crosslinker
BACE
Necroptosis
GTPase
c-Myc
Cysteine Protease
Liver X Receptor
Glucokinase
ABC Transporter
Fatty Acid Synthase
Hedgehog/Smoothened
PDGFR
CaMK
Survivin
Free radical scavengers
PAI-1
GST
Retinoid Receptor
Phospholipase
FGFR
MEK
Syk
c-Kit
DNA Methyltransferase
FAK
AhR
PKM
FOXO3
PGK1
GPCR
Chloride channel
Proton pump
PROTACs
CAT
Monocarboxylate transporter
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RAR/RXR
CD38
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gp120/CD4
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Adenylate cyclase
RIP kinase
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PAK
Bradykinin Receptor
PTEN
Somatostatin
Epoxide Hydrolase
Aurora Kinase
cAMP
glycosidase
DNA
SGLT
Beta-Secretase
PGE Synthase
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Acyltransferase
STING
LRRK2
Trk receptor
Urea Transporter
AIM2
transporter
ASK
Casein Kinase
RSV
ATM/ATR
Acetyl-CoA Carboxylase
p62
c-Fms
Protease
PDK
Aquaporin
Hydroxylase
FOXO
PLK
Cuproptosis
Complement System
Gap Junction Protein
DAPK
Platelet aggregation
IRAK
S6 Kinase
Sigma receptor
Thrombin
Lysosomal Autophagy
CFTR
MLK
PD-1/PD-L1
HER

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