购物车
0

抑制剂库
TargetMol

Inhibitor Library

细胞信号控制细胞基本活动,调控细胞行为。细胞感知并准确响应微环境的变化是发育、组织修复和免疫的基础,也是正常组织稳态的基础。细胞信号间相互作用异常或细胞信息处理错误是导致癌症、自身免疫和糖尿病等疾病的原因。深入了解细胞信号传导,疾病可得到更有效的治疗。

TargetMol 抑制剂库是由9730 个靶向小分子化合物组成的集合,每一个化合物都有明确的抑制靶点,靶点所处的信号通路也因此被阻断,TargetMol 抑制剂库是研究信号通路及相关疾病的有力工具,可用于高通量筛选和高内涵筛选。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L2000
产品编号: L2000
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
验证码

技术资料

产品描述
  • 产品描述:
    • 9730个小分子抑制剂的独特集合,主要用于细胞信号研究、新药筛选、高通量筛选和高内涵筛选;
    • 通过临床前研究和临床实验,生物活性和安全性已经得到验证;部分抑制剂已经被FDA批准上市;
    • 作用于MAPK、PI3K、JAK、HDAC、VEGFR、CDK等靶点,阻断相关信号通路;
    • 结构多样,药效显著,可渗透细胞;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
化合物库定制
我们的化合物库可以灵活定制! 了解更多>
您可以通过点击按钮
定制您专属的化合物!
化合物库组成
Apoptosis
Others
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
Parasite
Adrenergic Receptor
EGFR
Ras
Calcium Channel
HIV Protease
AChR
Dopamine Receptor
VEGFR
PDE
Dehydrogenase
Potassium Channel
ROS
Cytochromes P450
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Histone Methyltransferase
p38 MAPK
HDAC
Antifungal
ERK
Phosphatase
Akt
mTOR
JAK
Virus Protease
SARS-CoV
Src
FLT
Cholinesterase (ChE)
Microtubule Associated
Influenza Virus
STAT
Wnt/beta-catenin
TNF
iGluR
PARP
Reactive Oxygen Species
PDGFR
TRP/TRPV Channel
Topoisomerase
Prostaglandin Receptor
FGFR
GSK-3
Caspase
Interleukin
PKC
Raf
Bcl-2 Family
NO Synthase
HCV Protease
c-Kit
Monoamine Oxidase
Proteasome
MMP
GABA Receptor
c-Met/HGFR
RAAS
JNK
MAO
Ferroptosis
Bcr-Abl
Lipoxygenase
TGF-beta/Smad
ALK
MAPK
HSP
Phospholipase
Transferase
Adenosine Receptor
NMDAR
E1/E2/E3 Enzyme
DUB
GluR
Histone Demethylase
PPAR
Drug Metabolite
Beta Amyloid
Tyrosinase
Aurora Kinase
Serine Protease
GPCR
Integrin
ROCK
Kras
Serotonin Transporter
HIF/HIF Prolyl-Hydroxylase
Reductase
PKA
Tyrosine Kinases
Casein Kinase
AMPK
Anti-infection
CCR
MDM-2/p53
Mitochondrial Metabolism
MEK
IL Receptor
IκB/IKK
ATPase
Serine/threonin kinase
HSV
Reverse Transcriptase
Carbonic Anhydrase
Angiotensin-converting Enzyme (ACE)
Nucleoside Antimetabolite/Analog
P-gp
Mitophagy
Estrogen Receptor/ERR
HBV
IGF-1R
Androgen Receptor
Antiviral
Cysteine Protease
Sirtuin
CXCR
TLR
RIP kinase
Glucosidase
Histone Acetyltransferase
Proton pump
Antioxidant
Acyltransferase
c-RET
DNA-PK
CaMK
TAM Receptor
glycosidase
S6 Kinase
FAK
Leukotriene Receptor
Gamma-secretase
Norepinephrine
NOD-like Receptor (NLR)
NOS
LPL Receptor
P2X Receptor
Trk receptor
c-Fms
HIF
Estrogen/progestogen Receptor
PERK
ATM/ATR
Cannabinoid Receptor
Hedgehog/Smoothened
FAAH
NADPH
Immunology/Inflammation related
Opioid Receptor
Chk
Nrf2
DPP-4
Fatty Acid Synthase
PLK
HER
Kinesin
Neurokinin receptor
Syk
IDO
Glucocorticoid Receptor
Indoleamine 2,3-Dioxygenase (IDO)
p53
DYRK
Lipase
Pim
NOD
Endothelin Receptor
HMG-CoA Reductase
PD-1/PD-L1
Chloride channel
Glutathione Peroxidase
Antifection
transporter
PDK
DNA Methyltransferase
Smo
Xanthine Oxidase
SGLT
Aryl Hydrocarbon Receptor
Hydroxylase
IRAK
Thrombin
LTR
Rho
MAGL
LRRK2
Sigma receptor
ROS Kinase
YAP
P2Y Receptor
c-Myc
Glutaminase
BTK
Isocitrate Dehydrogenase (IDH)
PAK
DHFR
Factor Xa
Stearoyl-CoA Desaturase (SCD)
PGE Synthase
S1P Receptor
Mdm2
Amino Acids and Derivatives
IAP
cAMP
Retinoid Receptor
MRP
Cholecystokinin Receptor
Antifolate
Myosin
OX Receptor
Epoxide Hydrolase
Aminopeptidase
PI4K
BACE
Glucokinase
IRE1
Beta-Secretase
LPA Receptor
Complement System
Monocarboxylate transporter
CSF-1R
Monoamine Transporter
Neuropeptide Y Receptor
OXPHOS
Ephrin Receptor
RSV
GTPase
Telomerase
Lipid
PAI-1
Aromatase
ribosome
AhR
Ligands for Target Protein for PROTAC
DNA
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Dynamin
Tie-2
Adenylate cyclase
PAFR
ABC Transporter
GST
CFTR
MLK
ADC Cytotoxin
MicroRNA
Necroptosis
GRK
Vasopressin Receptor
STING
Acetyl-CoA Carboxylase
Platelet aggregation
NADPH-oxidase
MIF
DNA gyrase
Molecular Glues
Bradykinin Receptor
OAT
MNK
Pyroptosis
Neprilysin
Melanocortin Receptor
CRM1
MyD88
Na+/Ca2+ Exchanger
GNRH Receptor
LIM Kinase
Neurotensin Receptor
NAMPT
PYK2
FLAP
UGT
Glucagon Receptor
GlyT
Wee1
Porcupine
Methionine Adenosyltransferase (MAT)
Carboxypeptidase
SGK
p97
Prolyl Endopeptidase (PREP)
SIK
Phosphorylase
IKZF
PAD
ATP Citrate Lyase
ASK
CRFR
CGRP Receptor
Gap Junction Protein
DAPK
APC/C
MTP
PROTACs
IFNAR
Bcl-6
LDLR
LDL
Arp2/3 Complex
Ligands for E3 Ligase
DNA Alkylation
PTEN
cGAS
GPX
Protease
ROR
DNA Alkylator/Crosslinker
Arrestin
Progesterone Receptor
Melatonin Receptor
AAK1
Guanylate cyclase
MELK
Hippo pathway
Aquaporin
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
MALT
NEDD8
DprE1
Succinate Receptor 1 (SUCNR1)
CETP
Galectin
CaSR
ATG
Liver X Receptor
FXR
NR4A
Amylase
MTH1
MT Receptor
HCN Channel
Bombesin Receptor
CD73
Decarboxylase
KLF
CRISPR/Cas9
Oxytocin Receptor
FOXO
Adenosine Deaminase
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
ASBT
TOPK
VDAC
Vitamin
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Hexokinase
ACK1
Orphan Receptor
p62
FKBP
Imidazoline Receptor
PKM
Apelin receptor
CAT
Transaminase
Arginase
Factor VIIa
ASCT
Hck
Endonuclease
FABP
Haspin Kinase
PROTAC Linker
Somatostatin
KSP
Cadherin
GPCR19
AIM2
TSH Receptor
HuR
GHSR
Ferroportin
PGK1
GSNOR
NUDIX hydrolase
EBI2/GPR183
Y Box Binding Protein 1
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
Photosensitizer
RANKL/RANK
Annexin A
Neuropeptide FF Receptor
Integrase
Transketolase
Huntingtin
PSMA
Urea Transporter
hCE
PARG(Poly(ADP-ribose) Glycohydrolase)
Drug-Linker Conjugates for ADC
FOXO3
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Aconitase
Neuropeptide W
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Target Protein Ligand-Linker Conjugates
Stemness kinase
LAG-3
Photosystem (PS)
Adiponectin Receptor
Fas/FasL
PACAP
Anion Exchanger
Thioredoxin
Mucin
Glutathione reductase
MRGPR
Early 2 Factor (E2F)
E3 Ligase Ligand-Linker Conjugates
CD74
CPT
GluCls
NEDD4-1
Cuproptosis
REV-ERB
Fer/FerT kinase
Tight Junction Protein
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α

寻找合适的化合物库

您无法确定哪种化合物库最适合您的项目?或者您需要定制解决方案?Anymole随时为您提供帮助。
电话:400820-0310
合作:info@screeningcompound.com
技术支持:tech@screeningcompound.com
客服:service@screeningcompound.com
TargetMol | Target Loading
正在加载 ~