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代谢化合物库
TargetMol

Metabolism Compound Library

代谢是生物体内发生的用于维持生命的一系列有序化学反应的总称。这些反应使得生物体能够生长、繁殖以及对外界环境做出反应。代谢通常分为两类:分解代谢和合成代谢;分解代谢又称为异化作用,可以将环境中或细胞存储的营养物质进行分解以获得能量;合成代谢又称为同化作用,可以利用能量来合成细胞中的各个组分,二者的平衡使生物体保持自身的稳定,以适应环境。代谢中的化学反应几乎都是在酶的催化下进行的,从一个代谢物到另一个代谢物的代谢过程是通过一系列连续的酶促反应实现的,这种连续的酶促反应称为代谢途径。代谢紊乱、机体代谢途径的失调或中断会引发一系列代谢相关疾病。如糖尿病、肥胖、高血压、心血管疾病、癌症等。
Targetmol 代谢化合物库收集了3059 种代谢途径相关的化合物,是研究代谢相关疾病有用的工具。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L2560
产品编号: L2560
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 特点:
    • 3059种代谢途径相关生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
    • 靶向糖代谢、脂质代谢、核苷酸代谢等多个代谢途径;靶点包括GLUT、Hexokinase、Pyruvate Kinase;ATGL、MAGL、FAAH等代谢相关热门靶点;
    • 结构多样,药效显著,可渗透细胞;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 优势介绍:

    靶向脂代谢、糖代谢、核苷酸代谢、线粒体代谢等代谢通路相关靶点。

     Metabolism Compound Library
    注:仅分析分布数量大于等于10个以上的通路。

    涉及靶点相关性高,靶点数量多,包括Fatty Acid Synthase、Lipoxygenase、Mitochondrial Metabolism、α-glucosidase等。

     Metabolism Compound Library
    注:仅分析分布数量大于等于20个以上的靶点。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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