购物车
0

多靶点化合物库
TargetMol

Multi-Target Compound Library

复杂疾病的发病机制往往涉及多个生物靶点和信号通路的共同作用,单靶点药物可能难以达到理想的治疗效果。因此,单靶点治疗策略在某些情况下可能疗效有限。多靶点药物则能够同时作用于多个关键靶点或相关信号通路,产生协同效应,从而显著提高治疗效果。这种综合干预方式不仅有助于更全面地调控疾病相关的生物网络,还能有效降低因单一靶点突变而引发的耐药性风险。此外,由于不同靶点之间的协同作用,多靶点药物可在保证疗效的前提下减少药物使用剂量,进而降低毒副作用,提升药物治疗的安全性和耐受性。因此,多靶点药物为复杂疾病的治疗提供了更为系统和高效的策略。
TargetMol多靶点药物库收集了5200中多靶点化合物,靶向两个及以上不同靶点,可用于多靶点药物开发。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L9510
产品编号: L9510
  • 规格
  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
验证码

技术资料

产品描述
  • 产品描述:
    • TargetMol提供5200种多靶点化合物,可用于高通量筛选和高内涵筛选;
    • 部分化合物已经过FDA批准上市;
    • 结构多样,具有药用活性,可透过细胞;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR和HPLC检测技术保证产品高纯度;
    • 所有化合物现货供应。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
化合物库定制
我们的化合物库可以灵活定制! 了解更多>
您可以通过点击按钮
定制您专属的化合物!
化合物库组成
Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
NF-κB
Antibacterial
ROS
CDK
PI3K
COX
Dopamine Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Potassium Channel
AChR
EGFR
VEGFR
HIV Protease
Akt
Cytochromes P450
ERK
Reactive Oxygen Species
Calcium Channel
Antibiotic
p38 MAPK
TNF
Parasite
Ras
mTOR
Histamine Receptor
Caspase
Epigenetic Reader Domain
Sodium Channel
PPAR
JAK
Interleukin
Src
Others
Virus Protease
NO Synthase
Estrogen/progestogen Receptor
PDGFR
FLT
Ferroptosis
iGluR
PDE
STAT
Dehydrogenase
Bcl-2 Family
SARS-CoV
HDAC
FGFR
IL Receptor
Influenza Virus
Wnt/beta-catenin
PKC
Histone Methyltransferase
Estrogen Receptor/ERR
TRP/TRPV Channel
PARP
c-Kit
JNK
GSK-3
AMPK
GABA Receptor
MMP
Microtubule Associated
Antifungal
c-Met/HGFR
NMDAR
Bcr-Abl
Cholinesterase (ChE)
TLR
MDM-2/p53
GluR
Prostaglandin Receptor
Raf
ALK
MAPK
Phosphatase
MAO
HSV
Monoamine Oxidase
TGF-beta/Smad
Beta Amyloid
Mitophagy
Tyrosine Kinases
HIF/HIF Prolyl-Hydroxylase
Aurora Kinase
Topoisomerase
Drug Metabolite
HCV Protease
Proteasome
HSP
GPCR
MEK
PKA
P-gp
Nrf2
Casein Kinase
Cannabinoid Receptor
Lipoxygenase
Reverse Transcriptase
ATPase
Serotonin Transporter
E1/E2/E3 Enzyme
Norepinephrine
p53
Adenosine Receptor
Mitochondrial Metabolism
Sirtuin
IκB/IKK
ROCK
IGF-1R
LPL Receptor
RAAS
S6 Kinase
NOS
Antiviral
Phospholipase
Anti-infection
Serine Protease
TAM Receptor
HBV
Glucocorticoid Receptor
Gamma-secretase
DNA-PK
Opioid Receptor
Trk receptor
Retinoid Receptor
HIF
S1P Receptor
Carbonic Anhydrase
Serine/threonin kinase
Nucleoside Antimetabolite/Analog
c-RET
NOD-like Receptor (NLR)
HER
Integrin
Antioxidant
DUB
Androgen Receptor
Cysteine Protease
Histone Acetyltransferase
Tyrosinase
FAK
CaMK
c-Fms
PROTACs
Histone Demethylase
Progesterone Receptor
Mdm2
PERK
NOD
Transferase
DYRK
Pim
Rho
CXCR
HMG-CoA Reductase
Hedgehog/Smoothened
CCR
Angiotensin-converting Enzyme (ACE)
ATM/ATR
ROS Kinase
DNA Alkylator/Crosslinker
Reductase
Glutathione Peroxidase
RIP kinase
transporter
Syk
BACE
MRP
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
Glucosidase
Chk
Beta-Secretase
PLK
DNA Methyltransferase
Sigma receptor
KRas
NADPH
Antifection
Proton pump
IDO
P2X Receptor
Smo
DPP-4
Fatty Acid Synthase
Indoleamine 2,3-Dioxygenase (IDO)
Chloride channel
c-Myc
PAK
FAAH
Acyltransferase
AhR
Leukotriene Receptor
DNA Alkylation
DNA
CSF-1R
IAP
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
cAMP
glycosidase
SGLT
GPCR19
PDK
Kinesin
ADC Cytotoxin
YAP
LTR
Liver X Receptor
FXR
ABC Transporter
IRAK
Thrombin
P2Y Receptor
Melatonin Receptor
LDL
PGE Synthase
Amino Acids and Derivatives
IFNAR
Tie-2
UGT
PTEN
Telomerase
Lipid
MNK
Pyroptosis
LPA Receptor
Discoidin Domain Receptor (DDR)
PD-1/PD-L1
DHFR
Necroptosis
Myosin
MT Receptor
Molecular Glues
Endothelin Receptor
OX Receptor
OXPHOS
BCRP
LRRK2
PI4K
CFTR
BTK
GTPase
Antifolate
LIM Kinase
PYK2
DNA gyrase
Xanthine Oxidase
Epoxide Hydrolase
ribosome
Aromatase
MLK
Thyroid hormone receptor(THR)
MicroRNA
ROR
Ligands for Target Protein for PROTAC
Lipase
Adenylate cyclase
Annexin A
PAFR
Monoamine Transporter
Vasopressin Receptor
STING
Free radical scavengers
Aminopeptidase
Ephrin Receptor
RSV
GST
SGK
NADPH-oxidase
Arginase
SIK
Glucagon Receptor
Guanylate cyclase
Survivin
PAI-1
FKBP
CRISPR/Cas9
Hydroxylase
Complement System
Neurokinin receptor
Platelet aggregation
IKZF
RAR/RXR
MyD88
Arrestin
Factor Xa
NAMPT
Glucokinase
Glutaminase
IRE1
Phosphorylase
MAGL
Cadherin
ATP Citrate Lyase
OAT
ASK
GPX
Protease-activated Receptor
Imidazoline Receptor
NPC1L1
Dynamin
Na+/Ca2+ Exchanger
Bcl-6
AAK1
NR4A
MTH1
GRK
ACK1
Porcupine
AIM2
Decarboxylase
cGAS
Carboxypeptidase
FOXO
Melanin-concentrating Hormone Receptor (MCHR)
Transaminase
NEDD8
TOPK
OCT
Cholecystokinin Receptor
Hck
ATG
RANKL/RANK
Amylase
GlyT
Hexokinase
Ligands for E3 Ligase
Bombesin Receptor
PAD
Thrombopoietin Receptor
Wee1
GluCls
CRFR
Methionine Adenosyltransferase (MAT)
Melanocortin Receptor
GHSR
Aquaporin
Adenosine Deaminase
CGRP Receptor
Cuproptosis
Gap Junction Protein
FOXO3
Advanced Glycation End Products
Monocarboxylate transporter
CRM1
gp120/CD4
MIF
VDA
GNRH Receptor
ASCT
Cell Cycle Arrest
LDLR
FLAP
Neuropeptide FF Receptor
Adiponectin Receptor
FABP
Haspin Kinase
AAK1 (AP2 associated kinase 1)
Arp2/3 Complex
Na-K-Cl cotransporter
PROTAC Linker
KSP
Orphan Receptor
Huntingtin
Glutathione reductase
CPT
MELK
Hippo pathway
Neprilysin
p62
Protease
KLF
Oxytocin Receptor
REV-ERB
DAPK
BMI-1
Lysosomal Autophagy
PKM
Taste receptor
CAT
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
Aconitase
Cell wall
CETP
N-Acetylglucosaminyltransferase
CaSR
Photosensitizer
Prolyl Endopeptidase (PREP)
Fas/FasL
Anion Exchanger
Integrase
HCN Channel
Neuropeptide Y Receptor
Somatostatin
Urea Transporter
CD74
hCE
Acetyl-CoA Carboxylase
RXFP receptor
ATTECs
APC/C
Tight Junction Protein
p97

寻找合适的化合物库

您无法确定哪种化合物库最适合您的项目?或者您需要定制解决方案?Anymol随时为您提供帮助。
电话:400-820-0310
合作:info@screeningcompound.com
技术支持:tech@screeningcompound.com
客服:service@screeningcompound.com
TargetMol | Target Loading
正在加载 ~