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神经递质受体化合物库
TargetMol

Neurotransmitter Receptor Compound Library

神经递质是人类行为的化学基础。研究证实行为病理大都由一个或数个神经递质缺失或增多失平衡引起。躯体疾病也可由于特殊的神经径路障碍引起,例如帕金森病(PD)。脑内神经递质分为生物原胺类、氨基酸类、肽类、乙酰胆碱类等。生物原胺类神经递质包括:多巴胺(DA)、去甲肾上腺素(NE)、肾上腺素(E)、5-羟色胺(5-HT)也称(血清素)。氨基酸类神经递质包括:γ-氨基丁酸(GABA)、甘氨酸、谷氨酸、组胺。肽类神经递质分为:内源性阿片肽、P 物质、神经加压素、胆囊收缩素(CCK)、生长抑素、血管加压素和缩宫素、神经肽 Y。其它神经递质还有:核苷酸类、花生酸碱、阿南德酰胺、sigma 受体(σ受体)。在突触后膜或效应器细胞膜上有能与神经递质相结合的特殊蛋白质,称神经递质受体或突触后受体。许多精神药物作用于神经递质受体。

TargetMol 收集了 2120 种神经递质受体相关的化合物,可用于神经系统药物的开发。

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L2610
产品编号: L2610
  • 规格
  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
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技术资料

产品描述
  • 产品描述:
    • 2120种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
    • 靶点包括5-HT receptor、AChR、GABA receptor、dopamine receptor、Opiod receptor等;
    • 结构多样,药效显著,可渗透细胞;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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化合物库组成
5-HT Receptor
AChR
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
GABA Receptor
iGluR
GluR
Endogenous Metabolite
Adenosine Receptor
NMDAR
Apoptosis
Opioid Receptor
Autophagy
Cannabinoid Receptor
Others
Antibacterial
Norepinephrine
Serotonin Transporter
Calcium Channel
Potassium Channel
P2X Receptor
Neurokinin receptor
Cholinesterase (ChE)
Sodium Channel
Cytochromes P450
Parasite
ERK
ROS
P2Y Receptor
NF-κB
Akt
PDE
Drug Metabolite
Sigma receptor
TRP/TRPV Channel
Influenza Virus
TNF
Antibiotic
Interleukin
Reactive Oxygen Species
Caspase
HIV Protease
Beta Amyloid
SARS-CoV
DNA/RNA Synthesis
GPCR
Adenylate cyclase
Antifungal
Mitophagy
Virus Protease
PI3K
p38 MAPK
Ferroptosis
HDAC
VEGFR
Dehydrogenase
CaMK
COX
Bcl-2 Family
Histone Methyltransferase
PPAR
HCV Protease
P-gp
NO Synthase
PKC
Anti-infection
Monoamine Oxidase
MAO
cAMP
Lipoxygenase
Monoamine Transporter
mTOR
MMP
GSK-3
Phospholipase
Microtubule Associated
PERK
Nucleoside Antimetabolite/Analog
ABC Transporter
Hydroxylase
Imidazoline Receptor
PAFR
Gamma-secretase
Mitochondrial Metabolism
Angiotensin-converting Enzyme (ACE)
Trk receptor
Arrestin
TLR
RAAS
Epigenetic Reader Domain
Acyltransferase
AMPK
BACE
EGFR
MDM-2/p53
Transaminase
MRP
Antioxidant
HBV
Wnt/beta-catenin
FAAH
HSV
CCR
Amino Acids and Derivatives
Immunology/Inflammation related
IL Receptor
HIF/HIF Prolyl-Hydroxylase
Phosphatase
Melatonin Receptor
Leukotriene Receptor
Prostaglandin Receptor
Tyrosinase
JNK
PKA
Beta-Secretase
FOXO
Transferase
Glucocorticoid Receptor
transporter
STAT
DYRK
PARP
Platelet aggregation
IRAK
ROS Kinase
Aurora Kinase
HMG-CoA Reductase
Sirtuin
MAPK
RSV
Ras
Chloride channel
NOS
Aryl Hydrocarbon Receptor
Nrf2
GluCls
Integrin
CDK
Glucosidase
TGF-beta/Smad
NADPH
Necroptosis
GRK
MT Receptor
MEK
c-Met/HGFR
Na+/Ca2+ Exchanger
GTPase
Progesterone Receptor
c-Myc
CaSR
Rho
Liver X Receptor
HCN Channel
GST
Carboxypeptidase
Reverse Transcriptase
Gap Junction Protein
NOD
Estrogen/progestogen Receptor
MIF
Antifolate
Glutaminase
RIP kinase
Bcr-Abl
GlyT
Antifection
Fatty Acid Synthase
PAD
Androgen Receptor
Indoleamine 2,3-Dioxygenase (IDO)
FGFR
FAK
ATPase
Carbonic Anhydrase
LTR
NR4A
IAP
Adiponectin Receptor
glycosidase
DNA
ATP Citrate Lyase
CRISPR/Cas9
MicroRNA
Lipase
Syk
Monocarboxylate transporter
FXR
Topoisomerase
LDL
CXCR
PTEN
Pyroptosis
p53
Melanin-concentrating Hormone Receptor (MCHR)
Thyroid hormone receptor(THR)
Reductase
Hedgehog/Smoothened
JAK
IκB/IKK
ATM/ATR
Adenosine Deaminase
OCT
IDO
Annexin A
Raf
Na-K-Cl cotransporter
Bombesin Receptor
Stearoyl-CoA Desaturase (SCD)
ACK1
SGLT
Lipid
FLT
DNA Methyltransferase
S6 Kinase
NOD-like Receptor (NLR)

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