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非甾体类抗炎化合物库
TargetMol

Nonsteroidal Anti-Inflammatory Compound Library

非甾体抗炎药(Nonsteroidal Antiinflammatory Drugs,NSAIDs)是一类不含皮质激素甾体结构的抗炎药,NSAIDs 自阿司匹林于1898年首次合成后,100多年来已有百余种上千个品牌上市,这类药物包括阿司匹林、对乙酰氨基酚、吲哚美辛、萘普生、萘普酮、双氯芬酸、布洛芬、尼美舒利、罗非昔布、塞来昔布等,该类药物通过抑制环氧化酶、减少前列腺素的合成,从而发挥抗炎、抗风湿、止痛、退热和抗凝血等作用,在临床上广泛用于骨关节炎、类风湿性关节炎、多种发热和各种疼痛症状的缓解。

TargetMol 非甾体类抗炎化合物库收集了609 种非甾体类的抗炎相关化合物,可用于抗炎相关的药理研究和药物开发。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L4710
产品编号: L4710
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 产品描述:
    • 609种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
    • 包含常见非甾体抗炎药活性成分,如阿司匹林、吲哚美辛、舒林酸、布洛芬、吡罗昔康等;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR和HPLC技术保证产品高纯度。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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