购物车
0

核受体化合物库
TargetMol

Nuclear Receptor Compound Library

核受体是细胞内一类区别于膜受体的蛋白,它们与相应配体结合后,能够直接与基因组DNA 结合并调节相邻基因表达,因此这类受体被归类为转录因子。核受体在胚胎发育和机体内环境平衡中发挥关键作用。近年来,核受体家族在代谢性疾病领域受到广泛的关注,已有研究证明,它们与糖尿病、脂肪肝等疾病的发生发展密切相关,也被称为代谢性核受体。

TargetMol 汇集了755 种有文献报道的核受体相关化合物,适用于核受体相关信号通路及疾病研究,可用于高通量筛选和高内涵筛选。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L1510
产品编号: L1510
  • 规格
  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
验证码

技术资料

产品描述
  • 产品描述:
    • 755个核受体作用化合物的独特集合,可用于高通量筛选和高内涵筛选;
    • 提供产品的来源、化学信息和生物学信息,为筛选提供理论方向和研究基础;
    • 结构多样,药效显著,可渗透细胞;
    • NMR和HPLC技术保证产品高纯度。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
化合物库定制
我们的化合物库可以灵活定制! 了解更多>
您可以通过点击按钮
定制您专属的化合物!
化合物库组成
PPAR
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
Androgen Receptor
Glucocorticoid Receptor
Others
Apoptosis
Autophagy
Endogenous Metabolite
Antibacterial
ROS
Thyroid hormone receptor(THR)
Retinoid Receptor
FXR
NF-κB
Liver X Receptor
ROR
Progesterone Receptor
COX
Interleukin
Cytochromes P450
Reactive Oxygen Species
Akt
ERK
Drug Metabolite
Antifungal
Prostaglandin Receptor
NR4A
AMPK
Caspase
TNF
NO Synthase
p38 MAPK
Ferroptosis
JNK
IL Receptor
PROTACs
PI3K
Parasite
MMP
Antibiotic
Antioxidant
Nrf2
Potassium Channel
REV-ERB
RAR/RXR
GSK-3
Wnt/beta-catenin
Bcl-2 Family
STAT
GPCR
Dehydrogenase
Reductase
Phosphatase
Mitophagy
Calcium Channel
TRP/TRPV Channel
PKC
TGF-beta/Smad
HSP
SARS-CoV
GPCR19
Influenza Virus
AChR
Tyrosinase
HIV Protease
NOS
Adrenergic Receptor
Annexin A
PDE
CDK
Fatty Acid Synthase
mTOR
TLR
Sirtuin
GABA Receptor
ADC Cytotoxin
Virus Protease
PARP
VEGFR
Glucosidase
Antifection
Lipoxygenase
glycosidase
IGF-1R
CaMK
transporter
Phospholipase
Cannabinoid Receptor
Ras
HIF/HIF Prolyl-Hydroxylase
p53
Src
Integrin
Ligands for Target Protein for PROTAC
RAAS
Glutathione Peroxidase
c-Myc
MRP
HBV
iGluR
FABP
Gamma-secretase
ABC Transporter
Smo
JAK
Cholinesterase (ChE)
Angiotensin-converting Enzyme (ACE)
Epigenetic Reader Domain
Orphan Receptor
EGFR
DNA/RNA Synthesis
LRRK2
Histone Acetyltransferase
IκB/IKK
Acetyl-CoA Carboxylase
Aromatase
5-HT Receptor
FOXO
Complement System
MDM-2/p53
Anti-infection
DNA Methyltransferase
Sodium Channel
Microtubule Associated
FAK
AhR
FOXO3
Proteasome
ATPase
MicroRNA
Carbonic Anhydrase
Histone Methyltransferase
HCV Protease
MyD88
c-Met/HGFR
IFNAR
BACE
Arrestin
Histone Demethylase
PERK
gp120/CD4
Melatonin Receptor
GNRH Receptor
PKA
Photosensitizer
Serine Protease
Cysteine Protease
Leukotriene Receptor
Glucokinase
MAO
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
Prolyl Endopeptidase (PREP)
Topoisomerase
Adenylate cyclase
FLAP
UGT
LDL
Raf
Glucagon Receptor
Phosphorylase
Mitochondrial Metabolism
Opioid Receptor
Ligands for E3 Ligase
PAK
Bombesin Receptor
Hedgehog/Smoothened
HSV
Xanthine Oxidase
Epoxide Hydrolase
cAMP
GluR
DNA
Lipid
Huntingtin
PGE Synthase
PSMA
P-gp
Survivin
Ephrin Receptor
CPT
Pyroptosis
Beta Amyloid
FKBP
Kras
PDK
Hydroxylase
FGFR
MEK
Gap Junction Protein
FLT
Syk
c-Kit
BMI-1
NOD
HMG-CoA Reductase
Sigma receptor
TAM Receptor
Thrombin
Liposome
NOD-like Receptor (NLR)
S1P Receptor
Vitamin

寻找合适的化合物库

您无法确定哪种化合物库最适合您的项目?或者您需要定制解决方案?Anymol随时为您提供帮助。
电话:400-820-0310
合作:info@screeningcompound.com
技术支持:tech@screeningcompound.com
客服:service@screeningcompound.com
TargetMol | Target Loading
正在加载 ~