购物车
0

蛋白翻译后修饰化合物库
TargetMol

Post-Translational Modification Compound Library

蛋白翻译后修饰(Post-Translational Modification, PTM)是指蛋白质在合成后经历的一系列化学修饰过程,这些修饰能够显著改变蛋白质的结构、功能和定位,从而在细胞信号传导、代谢调控、应激反应等众多生物学过程中发挥关键作用。常见的翻译后修饰包括磷酸化、乙酰化、泛素化、糖基化等。研究发现,许多疾病的发生和发展与蛋白翻译后修饰的异常密切相关,例如癌症、神经退行性疾病(如阿尔茨海默病和帕金森病)、糖尿病以及心血管疾病等。因此,对蛋白翻译后修饰的研究不仅有助于揭示疾病机制,还为新药开发提供了重要的靶点。
TargetMol 翻译后修饰化合物库收集了3490种小分子活性化合物,该库涵盖了多种能够调控翻译后修饰酶活性的化合物,包括激酶、乙酰转移酶、泛素连接酶等相关靶点的调节剂。可广泛应用于信号通路机制研究、新靶点发现与验证、高通量药物筛选,是蛋白翻译后修饰研究和药物筛选的有效工具。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L1620
产品编号: L1620
  • 规格
  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
化合物库咨询特别折扣,等您来咨询!
验证码

技术资料

产品描述
  • 产品描述:
    • 收录了3490种小分子活性化合物,用于翻译后修饰相关研究;
    • 包含针对激酶、乙酰转移酶、泛素连接酶等蛋白翻译后修饰相关酶的调节剂;
    • 部分化合物已获美国食品药品监督管理局(FDA)批准;
    • 详细的说明书,化合物结构、靶点信息、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
化合物库定制
我们的化合物库可以灵活定制! 了解更多>
您可以通过点击按钮
定制您专属的化合物!
化合物库组成
Apoptosis
Autophagy
CDK
PI3K
EGFR
VEGFR
Histone Methyltransferase
p38 MAPK
HDAC
Akt
JAK
ERK
mTOR
Src
PARP
FLT
NF-κB
Others
PKC
PDGFR
AMPK
GSK-3
FGFR
Raf
c-Kit
c-Met/HGFR
Bcr-Abl
Endogenous Metabolite
ALK
MAPK
JNK
BTK
Antibacterial
Ras
Aurora Kinase
Histone Demethylase
PKA
Epigenetic Reader Domain
Casein Kinase
MEK
Caspase
ROS
Tyrosine Kinases
ROCK
Parasite
TGF-beta/Smad
E1/E2/E3 Enzyme
IκB/IKK
STAT
IGF-1R
Wnt/beta-catenin
Serine/threonin kinase
RIP kinase
Glucosidase
TNF
FAK
c-RET
CaMK
DNA-PK
Trk receptor
Histone Acetyltransferase
S6 Kinase
TAM Receptor
Bcl-2 Family
ATM/ATR
PERK
Glucokinase
c-Fms
DNA/RNA Synthesis
PLK
COX
HER
HIV Protease
glycosidase
Syk
Virus Protease
Interleukin
Mitophagy
Chk
Influenza Virus
PROTACs
DYRK
Pim
Serine Protease
Phosphatase
Reactive Oxygen Species
ROR
IRAK
Transferase
PPAR
Antibiotic
Potassium Channel
NO Synthase
PDK
Tyrosinase
PAK
LRRK2
Ferroptosis
IL Receptor
Cytochromes P450
ROS Kinase
Calcium Channel
Dehydrogenase
IRE1
PDE
Ephrin Receptor
MDM-2/p53
Adrenergic Receptor
HSV
MMP
AChR
Beta Amyloid
PI4K
5-HT Receptor
Antifungal
Nrf2
Adenosine Receptor
Microtubule Associated
Tie-2
CSF-1R
MNK
Antiviral
SARS-CoV
Sirtuin
Discoidin Domain Receptor (DDR)
MLK
Kras
YAP
Drug Metabolite
S1P Receptor
GRK
Wee1
HSP
Sodium Channel
Histamine Receptor
PYK2
Cholinesterase (ChE)
TLR
SGK
Anti-infection
p53
Kinesin
PKM
Mdm2
HCV Protease
Antioxidant
SIK
Mitochondrial Metabolism
PAD
P-gp
Monoamine Oxidase
Dopamine Receptor
Integrin
Ligands for Target Protein for PROTAC
LIM Kinase
MAO
Topoisomerase
Gamma-secretase
Antifection
Acyltransferase
GABA Receptor
DAPK
TOPK
AAK1
Rho
TRP/TRPV Channel
Aryl Hydrocarbon Receptor
Molecular Glues
Angiotensin-converting Enzyme (ACE)
transporter
MELK
IKZF
ATPase
NOS
MyD88
IFNAR
Necroptosis
Myosin
PTEN
Lipoxygenase
Prostaglandin Receptor
STING
ASK
Cannabinoid Receptor
HIF/HIF Prolyl-Hydroxylase
Carbonic Anhydrase
NEDD8
Estrogen/progestogen Receptor
LPL Receptor
RAAS
c-Myc
Estrogen Receptor/ERR
HBV
Hck
LDL
AAK1 (AP2 associated kinase 1)
Hexokinase
DNA Alkylation
ACK1
GluR
Hippo pathway
Carboxypeptidase
FKBP
NOD-like Receptor (NLR)
PD-1/PD-L1
BACE
NADPH
Cholecystokinin Receptor
Nucleoside Antimetabolite/Analog
FXR
NR4A
IDO
IAP
Haspin Kinase
Monoamine Transporter
Fatty Acid Synthase
Hedgehog/Smoothened
DUB
Indoleamine 2,3-Dioxygenase (IDO)
OXPHOS
BCRP
PAI-1
Pyroptosis
Reverse Transcriptase
Phospholipase
DNA Methyltransferase
NOD
GPCR
Proteasome
Chloride channel
Proton pump
GDNF
gp120/CD4
Glutathione Peroxidase
GTPase
Antifolate
Liver X Receptor
NAMPT
Amylase
Immunology/Inflammation related
iGluR
Glucagon Receptor
NMDAR
Cadherin
cAMP
ATP Citrate Lyase
Lipid
Beta-Secretase
Survivin
Porcupine
cGAS
Retinoid Receptor
FOXO3
CRISPR/Cas9
HIF
BMI-1
FOXO
ADC Cytotoxin
Apelin receptor
MicroRNA
NPC1L1
RAR/RXR
DHFR
Amino Acids and Derivatives
Y Box Binding Protein 1
Reductase
Progesterone Receptor
Melatonin Receptor
Bcl-6
MRP
ATG
Serotonin Transporter
Cell Cycle Arrest
Stemness kinase
Glutaminase
LDLR
RANKL/RANK
Prolyl Endopeptidase (PREP)
Adenylate cyclase
UGT
PAFR
P2X Receptor
Opioid Receptor
PROTAC Linker
Ligands for E3 Ligase
Bombesin Receptor
FAAH
CCR
CXCR
Thrombopoietin Receptor
Norepinephrine
DNA
Androgen Receptor
Telomerase
PGE Synthase
PSMA
Free radical scavengers
E3 Ligase Ligand-Linker Conjugates
Aminopeptidase
AIM2
Decarboxylase
RSV
NEDD4-1
Acetyl-CoA Carboxylase
p62
TMV
Protease
Aromatase
Hydroxylase
RXFP receptor
REV-ERB
Fer/FerT kinase
Gap Junction Protein
NADPH-oxidase
MAP3K
HMG-CoA Reductase
Sigma receptor
Protease-activated Receptor
p97
CFTR

寻找合适的化合物库

您无法确定哪种化合物库最适合您的项目?或者您需要定制解决方案?Anymol随时为您提供帮助。
电话:400-820-0310
合作:info@screeningcompound.com
技术支持:tech@screeningcompound.com
客服:service@screeningcompound.com
TargetMol | Target Loading
正在加载 ~