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酪氨酸激酶分子库
TargetMol

Tyrosine Kinase Inhibitor Library

蛋白激酶(PK)是正常细胞信号转导的重要介质,通过对底物蛋白的磷酸化来调节它们的活性、定位和整体功能。蛋白激酶参与几乎所有细胞过程的活动,在细胞增殖、血管生成、迁移、细胞周期等过程中发挥关键作用。在众多蛋白激酶中,酪氨酸蛋白激酶(TK)可能是癌症治疗较有吸引力的靶点,因为TK 信号异常通常与肿瘤发生发展密切相关,此外,TK 在炎症和类风湿性关节炎等其他疾病中也起着关键作用。

TargetMol 酪氨酸激酶分子库精选 1350 种酪氨酸激酶抑制剂,用于研究酪氨酸激酶相关的疾病和药物,可用于高通量筛选和高内涵筛选。

  • 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L2200
产品编号: L2200
  • 规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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技术资料

产品描述
  • 产品描述:
    • 1350种酪氨酸激酶抑制剂的独特集合,可用于高通量筛选和高内涵筛选;
    • 靶点含c-kit、c-Met、EGFR、FGFR、SRC、JAK、SYK、Btk、Bcr-Abl等;
    • 通过临床前研究和临床实验,生物活性和安全性已经得到验证,部分产品已被FDA批准上市;
    • 结构多样,药效显著,可渗透细胞;
    • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
    • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
  • 包装和储存:
    • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
    • 干粉蓝冰运输,DMSO溶液干冰运输;
    • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
    • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。
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