Name: MK-4256
Rating: 5 (10 reviews)

有库存

sdf 文件

结构编辑

类似物检索

HIT ID:HIT212672559
Cas No:1104599-69-0
常用名:MK-4256
IUPAC:3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrazol-4-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole
IUPAC:3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrazol-4-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole
InChI key:NTIFDLOQPKMIJK-AJTFRIOCSA-N

分子式:C27H23FN8O
分子量:494.534
氢键供体数 (HBD):3
氢键受体数 (HBA):5
LogP:3.501604
SMILES:Cc1nc(no1)[C@@]1(N[C@H](Cc2c1[nH]c1ccccc21)c1ncc([nH]1)-c1ccc(F)cc1)c1cnn(C)c1
SMILES:Cc1nc(no1)[C@@]1(N[C@H](Cc2c1[nH]c1ccccc21)c1ncc([nH]1)-c1ccc(F)cc1)c1cnn(C)c1

MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively).

市场产品/服务共显示1个结果

您无法确定哪种化合物库最适合您的项目？或者您需要定制解决方案？Anymole随时为您提供帮助。

电话：400820-0310

合作：info@screeningcompound.com

技术支持：tech@screeningcompound.com

客服：service@screeningcompound.com

正在加载 ~