Name: Zaldaride maleate
Rating: 5 (10 reviews)

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结构编辑

类似物检索

HIT ID:HIT212673535
Cas No:109826-27-9
常用名:Zaldaride maleate
别名:KW 5617, CGS-9343B
IUPAC:(2Z)-but-2-enedioic acid; 1-[1-({7-methyl-8-oxa-2-azatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,10,12-pentaen-7-yl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
IUPAC:(2Z)-but-2-enedioic acid; 1-[1-({7-methyl-8-oxa-2-azatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,10,12-pentaen-7-yl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
InChI key:NGODOSILXOFQPH-BTJKTKAUSA-N

分子式:C30H32N4O6
分子量:544.608
氢键供体数 (HBD):1
氢键受体数 (HBA):3
LogP:3.8678033
SMILES:OC(=O)\C=C/C(O)=O.CC1(CN2CCC(CC2)n2c3ccccc3[nH]c2=O)OCc2ccccc2-n2cccc12
SMILES:OC(=O)\C=C/C(O)=O.CC1(CN2CCC(CC2)n2c3ccccc3[nH]c2=O)OCc2ccccc2-n2cccc12

Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate is an effective and selective inhibitor of calmodulin. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+, and K+ currents in PC12 cells and inhibits nAChR.

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