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  3. HIT212713519
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HIT212713519
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HIT212713519
  • HIT ID:HIT212713519
  • Cas No:139088-45-2
  • 常用名:RP-72540
  • 别名:RPR-102681, RPR102681, RPR 102681
  • IUPAC:2-{3-[({[(3-methoxyphenyl)({[methyl(phenyl)carbamoyl]methyl})carbamoyl]methyl}carbamoyl)amino]phenyl}propanoic acid
    IUPAC:2-{3-[({[(3-methoxyphenyl)({[methyl(phenyl)carbamoyl]methyl})carbamoyl]methyl}carbamoyl)amino]phenyl}propanoic acid
  • InChI key:ZDOYTKRSYALDTJ-UHFFFAOYSA-N
  • 分子式:C28H30N4O6
  • 分子量:518.57
  • 氢键供体数 (HBD):3
  • 氢键受体数 (HBA):6
  • LogP:2.6768525
  • SMILES:COc1cccc(c1)N(CC(=O)N(C)c1ccccc1)C(=O)CNC(=O)Nc1cccc(c1)C(C)C(O)=O
    SMILES:COc1cccc(c1)N(CC(=O)N(C)c1ccccc1)C(=O)CNC(=O)Nc1cccc(c1)C(C)C(O)=O
  • RP-72540 is a cholecystokinin B receptor antagonist. RP 72540 showed selectivity factors in express of 200 for CCKA versus CCKB receptors and also had high affinity for gastrin binding sites in the stomach. Administration of RP-72540 resulted in a dose-dependent inhibition of [3H]pCCK-8 binding in mouse brain homogenate. However, the relative penetration of RP-72540 into the forebrain after peripheral administration was below 0.01%.
市场产品/服务共显示1个结果
  • 供应商
    TargetMolSC
    规格
    货期
    6-8周
    纯度
    -
    ¥ 10,600.00
    1

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