Name: TP-238 hydrochloride
Rating: 5 (10 reviews)

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结构编辑

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HIT ID:HIT214323465
Cas No:2415263-05-5
常用名:TP-238 hydrochloride
IUPAC:6-{4-[3-(dimethylamino)propoxy]phenyl}-2-methanesulfonyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-4-amine hydrochloride
IUPAC:6-{4-[3-(dimethylamino)propoxy]phenyl}-2-methanesulfonyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-4-amine hydrochloride
InChI key:FHVADRKEPFRFFF-UHFFFAOYSA-N

分子式:C22H31ClN6O3S
分子量:495.04
氢键供体数 (HBD):
氢键受体数 (HBA):
LogP:
SMILES:Cl.CN(C)CCCOc1ccc(cc1)-c1cc(NCCCn2cccn2)nc(n1)S(C)(=O)=O
SMILES:Cl.CN(C)CCCOc1ccc(cc1)-c1cc(NCCCn2cccn2)nc(n1)S(C)(=O)=O

TP-238 hydrochloride is a highly potent and selective dual CECR2/BPTF probe, demonstrating IC50 values of 30 nM and 350 nM, respectively. It additionally exerts inhibitory effects on BRD9, with a pIC50 value of 5.9, while displaying lower activity against 338 other kinases.

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