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- HIT ID:HIT214433658
- Cas No:1685235-41-9
- 常用名:Dyrk1A-IN-5
- InChI key:SDRAETFVRBBLOB-UHFFFAOYSA-N
- 分子式:C16H9IN2O2
- 分子量:388.164
- 氢键供体数 (HBD):
- 氢键受体数 (HBA):
- LogP:
- Dyrk1A-IN-5 (compound 5j) is a highly potent and selective inhibitor of DYRK1A, exhibiting an IC50 of 6 nM. It dose-dependently diminishes the phosphorylation of Thr434 in SF3B1, with an IC50 of 0.5 μM. Moreover, Dyrk1A-IN-5 effectively inhibits the phosphorylation of tau at Thr212, with an IC50 of 2.1 μM. Given these properties, Dyrk1A-IN-5 is a valuable tool for Down syndrome research [1].
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- 供应商TargetMol规格货期5日内发货纯度-¥ 2,180.001
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