Name: Desmethyl-YM-298198
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HIT ID:HIT218695663
Cas No:299901-57-8
Common Name:Desmethyl-YM-298198
IUPAC:11-amino-N-cyclohexyl-3-methyl-5-thia-2,7-diazatricyclo[6.4.0.0^{2,6}]dodeca-1(12),3,6,8,10-pentaene-4-carboxamide
IUPAC:11-amino-N-cyclohexyl-3-methyl-5-thia-2,7-diazatricyclo[6.4.0.0^{2,6}]dodeca-1(12),3,6,8,10-pentaene-4-carboxamide
InChI key:VWOMTTIMBHBPBI-UHFFFAOYSA-N

Molecular Formula:C17H20N4OS
Molecular Weight:328.43
Hydrogen Bond Donor (HBD):
Hydrogen Bond Acceptor (HBA):
LogP:
SMILES:Cc1c(sc2nc3ccc(N)cc3n12)C(=O)NC1CCCCC1
SMILES:Cc1c(sc2nc3ccc(N)cc3n12)C(=O)NC1CCCCC1

Desmethyl-YM-298198 is a highly affine, selective, non-competitive antagonist of mGluR1 (IC50: 16 nM). It demonstrates analgesic effects in mice with pain hypersensitivity induced by Streptozotocin.

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