Name: Salvinorin A Carbamate
Rating: 5 (10 reviews)

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HIT ID:HIT218832934
Cas No:
常用名:Salvinorin A Carbamate
别名:Sal A Carbamate, Divinorin A Carbamate
IUPAC:methyl 9-(carbamoyloxy)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-naphtho[2,1-c]pyran-7-carboxylate
IUPAC:methyl 9-(carbamoyloxy)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-naphtho[2,1-c]pyran-7-carboxylate
InChI key:FHTGZEVOZWRYEL-UHFFFAOYSA-N

分子式:C22H27NO8
分子量:433.457
氢键供体数 (HBD):
氢键受体数 (HBA):
LogP:
SMILES:COC(=O)C1CC(OC(N)=O)C(=O)C2C1(C)CCC1C(=O)OC(CC21C)c1ccoc1
SMILES:COC(=O)C1CC(OC(N)=O)C(=O)C2C1(C)CCC1C(=O)OC(CC21C)c1ccoc1

Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.

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