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Advanced Glycation End Products
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Targetmol为生命科学及医药领域的科研人员提供其他未细分细胞信号通路相关产品,包括抑制剂、激动剂、调节剂、降解剂等。
HIT212063045
1H-Pyrrolo[3,2-c]pyridin-4-amine
T67639
60290-23-5
1H-Pyrrolo[3,2-c]pyridin-4-amine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67639,CAS号为 60290-23-5。
Others
HIT217588509
Tolytoxin
T71063
127999-44-4
Tolytoxin is a cytostatic, antifungal macrolide produced by blue-green algae of the genus Scytonema, is a potent, reversible inhibitor of cytokinesis in cultured mammalian cells
Others
HIT101648727
5-Azauracil
TNU0814
71-33-0
Heterocyclic Compounds –Triazine; Intermediates and Building Blocks - Nucleophile; Nucleoside base
Others
HIT212724831
Hydroquinone monobenzoate
T71887
2444-19-1
Hydroquinone monobenzoate is an oxidoreductant and potential topoisomerase II inhibitor commercially used in skin whitening treatments and photography development. It may induce DNA damage.
Others
HIT214435863
N4-Benzoyl-1-(6-O-DMTr-2,3-dideoxy-beta-D-erythro-hexopyranosyl)cytosine
TNU1623
145594-00-9
N4-Benzoyl-1-(6-O-DMTr-2,3-dideoxy-beta-D-erythro-hexopyranosyl)cytosine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU1623,CAS号为 145594-00-9。
Others
HIT103895525
2-(2-Ethoxyphenoxy)ethanamine
T66134
6781-17-5
2-(2-Ethoxyphenoxy)ethanamine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66134,CAS号为 6781-17-5。
Others
HIT106881829
Methyl (4-chloro-3-(trifluoromethyl)phenyl)carbamate
T64807
Methyl (4-chloro-3-(trifluoromethyl)phenyl)carbamate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64807。
Others
HIT212000872
N-(2-(Diethylamino)ethyl)-5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxamide
T66203
356068-86-5
N-(2-(Diethylamino)ethyl)-5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66203,CAS号为 356068-86-5。
Others
HIT218850805
Malacidin A
T75528
2254483-95-7
Malacidin A 是一种钙依赖性抗生素。Malacidin A 对许多耐药病原体,特别是革兰氏阳性菌具有高度活性。
Others
HIT107740036
N-Phenylpropionamide
T66814
620-71-3
N-Phenylpropionamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66814,CAS号为 620-71-3。
Others
HIT214432894
2-Amino-4-chloro-5-iodo-N2-pivaloyl-7-[2-deoxy-3,5-di-O- (4-methylbenzoyl)-b-D-ribofuanosyl]-7H-pyrrolo[2,3-d]pyrimidine
TNU1291
199938-73-3
2-Amino-4-chloro-5-iodo-N2-pivaloyl-7-[2-deoxy-3,5-di-O- (4-methylbenzoyl)-b-D-ribofuanosyl]-7H-pyrrolo[2,3-d]pyrimidine is a Nucleoside Derivative - 7-Deazapurine nucleoside; Halo-nucleoside.
Others
HIT212032235
endo-Hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione
T66460
28871-95-6
endo-Hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66460,CAS号为 28871-95-6。
Others
HIT103822480
6,7-Dihydroxyquinazolin-4(3H)-one
T66641
16064-15-6
6,7-Dihydroxyquinazolin-4(3H)-one 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66641,CAS号为 16064-15-6。
Others
HIT212721470
5'-Deoxyuridine
TNU1184
15958-99-3
5'-Deoxyuridine is a Nucleoside Derivative - 5'-Modified nucleoside;5'-Deoxy nucleoside.
Others
HIT217590887
LY2457546
T68389
908265-94-1
LY2457546 is a potent and orally bioavailable inhibitor of multiple receptor tyrosine kinases involved in angiogenic and tumorigenic signalling. LY2457546 demonstrates potent activity against targets that include VEGFR2 (KDR), PDGFRβ, FLT-3, Tie-2 and members of the Eph family of receptors. In vivo, LY2457546 inhibited VEGF-driven autophosphorylation of lung KDR in the mouse and rat in a dose and concentration dependent manner. LY2457546 was well tolerated and exhibited efficacy in a 13762 syngeneic rat mammary tumor models. Additionally, LY2457546 caused complete regression of well-established tumors in an acute myelogenous leukemia (AML) FLT3-ITD mutant xenograft tumor model. The unique spectrum of target activity, potent in vivo anti-tumor efficacy in a variety of rodent and human solid tumor models, exquisite potency against a clinically relevant model of AML, and non-clinical safety profile justify the advancement of LY2457546 into clinical testing. (source: Invest New D......
Others
HIT214434422
2-Amino-6-chloro-9-(3-deoxy-2-O-acetyl-5-O-benzoyl-beta-D-ribofuanosyl)-9H-purine
TNU0982
2095417-15-3
2-Amino-6-chloro-9-(3-deoxy-2-O-acetyl-5-O-benzoyl-beta-D-ribofuanosyl)-9H-purine is a Nucleoside Derivative - 3'-Deoxy nucleoside, Halo-nucleoside; Scaffold and Template.
Others
HIT214458705
Nitrodenafil
T71937
147676-99-1
Nitrodenafil is a related compound of Sildenafil -- a phosphodiesterase inhibitor.
Others
HIT105226908
10,11-Dihydro-11-oxodibenzo[b,f][1,4]thiazepine
T65432
3159-07-7
10,11-Dihydro-11-oxodibenzo[b,f][1,4]thiazepine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65432,CAS号为 3159-07-7。
Others
HIT217589782
LC-1310
T69681
2322268-24-4
LC-1310 is an irreversible p97 inhibitor.
Others
HIT212040806
Boc-Asp(OAll)-OH
T66689
132286-77-2
Boc-Asp(OAll)-OH 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66689,CAS号为 132286-77-2。
Others
HIT104677562
2-(4-Isobutylphenyl)propanamide
T66977
2-(4-Isobutylphenyl)propanamide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T66977。
Others
HIT217585251
CYMAL-6 Neopentyl Glycol
TF0123
1423306-24-4
CYMAL-6 Neopentyl Glycol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0123,CAS号为 1423306-24-4。
Others
HIT214435878
2-Amino -7-propargyl-7,8-dihydro-8-oxo-9-(beta-D-2,3,5-tri-O-actyl-xylofuranosyl)purine
TNU1331
2389988-52-5
2-Amino -7-propargyl-7,8-dihydro-8-oxo-9-(beta-D-2,3,5-tri-O-actyl-xylofuranosyl)purine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU1331,CAS号为 2389988-52-5。
Others
HIT100421456
G-573
T71891
22868-35-5
G-573 is an allosteric inhibitor of MEK that is both potent and selective. The IC(50) value for pERK inhibition in HCT116 tumours by G-573 was estimated to be 0.406 µM. The IC(50) values for tumour growth inhibition in HCT116 and H2122 were estimated to be 3.43 and 2.56 µM, respectively. ED(50) estimates in HCT116 and H2122 mouse xenograft models were estimated to be ~4.6 and 1.9 mg/kg/day, respectively.
Others
HIT217589577
SAS-0132
T69920
2095551-89-4
SAS-0132 is a modulator/antagonist of sigma2R/TMEM97 and has potential for treating TBIs, Alzheimer's disease, and neuropathic pain.
Others
HIT217588861
NA 382
T70683
143086-33-3
NA 382 is a staurosporine derivative that inhibits multidrug resistance.
Others
HIT217590589
Cantharidin imide
T68721
76970-77-9
Cantharidin imide is a PP1/2A inhibitor found in Canarthis vesicatoria. It inhibits proliferation of colorectal cancer cells, increases MCP-1, IL-6, and IL-β levels, and inhibits differentiation and resorptive activity of osteoclasts. This compound can produce severe skin inflammation, and is extremely toxic if ingested orally.
Others
HIT105127275
4-Methoxy-2-nitroacetanilide
T67311
119-81-3
4-Methoxy-2-nitroacetanilide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67311,CAS号为 119-81-3。
Others
HIT212876315
D-(+)-Cellotriose
T65097
33404-34-1
(2R,3R,4R,5R)-4-(((2S,3R,4R,5S,6R)-3,4-Dihydroxy-6-(hydroxymethyl)-5-(((2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)oxy)tetrahydro-2H-pyran-2-yl)oxy)-2,3,5,6-tetrahydroxyhexanal 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T65097,CAS号为 33404-34-1。
Others
HIT212041943
NU1085
T71908
188106-83-4
NU1085 is a potent poly(ADP-ribose) polymerase (PARP) inhibitors have been developed that potentiate the cytotoxicity of ionizing radiation and anticancer drugs. The biological effects of NU1085 [Ki = 6 nM], in combination with temozolomide (TM) or topotecan (TP) have been studied in 12 human tumor cell lines (lung, colon, ovary, and breast cancer). Cells were treated with increasing concentrations of TM or TP +/- NU1085 (10 microM) for 72 h.
Others
HIT102948960
1-(2-Amino-4,5-dimethoxyphenyl)ethanone
T64852
4101-30-8
1-(2-Amino-4,5-dimethoxyphenyl)ethanone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64852,CAS号为 4101-30-8。
Others
HIT217590639
Ciladopa (free base)
T68676
80109-27-9
Ciladopa (free base) is a dopamine agonist with a similar chemical structure to dopamine. It was under investigation as an antiparkinsonian agent but was discontinued due to concerns of tumorogenesis in rodents.
Others
HIT106828076
Morpholin-4-yl-acetic acid
T65322
3235-69-6
Morpholin-4-yl-acetic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65322,CAS号为 3235-69-6。
Others
HIT214432765
Triclofos
T60297
306-52-5
Triclofos 是一种有效的口服活性的镇静剂。Triclofos 在体内可迅速水解成 trichloroethanol (TCEOH) 和磷酸一钠,有助于镇静。
Others
HIT217589094
Abivertinib HCl
T70446
1557268-90-2
Abivertinib, also known as AC0010 and Avitinib, is a third-generation EGFR tyrosine kinase inhibitor and BTK Inhibitor that demonstrated clinical efficacy and manageable adverse events (AEs). Abivertinib inhibits cell proliferation, reduces colony-forming capacity, and induces apoptosis and cell cycle arrest in AML cells, especially those harboring FLT3-ITD mutations. Abivertinib was also found to be more sensitive than ibrutinib in treating AML. Abivertinib may be a promising novel agent for AML, with potential for combination treatment with HHT.
Others
HIT214308524
(S)-2-((tert-Butoxycarbonyl)amino)-3-(2-methoxyphenyl)propanoic acid
T67248
(S)-2-((tert-Butoxycarbonyl)amino)-3-(2-methoxyphenyl)propanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67248。
Others
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