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供应商货号
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供应商货号
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化合物库
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Advanced Glycation End Products
CYP19A1
Decarboxylase
DprE1
Fer/FerT kinase
Platelet aggregation
Progesterone Receptor
Others
信号通路
其他
Others
Others
Targetmol为生命科学及医药领域的科研人员提供其他未细分细胞信号通路相关产品,包括抑制剂、激动剂、调节剂、降解剂等。
HIT214323066
Orexin 2 Receptor Agonist 2
T39561
2114324-60-4
Orexin 2 Receptor Agonist 2 (ORA-2) is a specific agonist for the orexin 2 receptor.
Others
OX Receptor
HIT212080452
Thalidomide-O-amido-PEG3-C2-NH2
T17915
1957236-20-2
Thalidomide-O-amido-PEG3-C2-NH2 (Cereblon Ligand-Linker Conjugates 3) is an E3 ligase ligand-linker conjugate which is designed using Thalidomide-based cereblon ligand and a 3-unit PEG linker. This compound is synthesized specifically for utilization in PROTAC technology.
Apoptosis
Autophagy
E3 Ligase Ligand-Linker Conjugates
Others
PROTAC Linker
HIT214323643
RM-018
T40269
2641993-55-5
RM-018 is a powerful tricomplex inhibitor that specifically targets the active state of KRAS G12C. It exhibits unique functional characteristics and possesses the ability to bind and inhibit both KRAS G12C and KRAS G12C/Y96D, potentially overcoming resistance.
Kras
Others
Ras
HIT212667767
Halo PROTAC 1
T17995
2241668-45-9
Halo PROTAC 1 is a PROTAC, which is a ligand having activity to bind to an intracellular proteins fused with HaloTag and a structure having activity to induce autophagy of an intracellular molecule are linked via a PEG linker[1].
AUTACs
Others
PROTACs
HIT218852367
AVE-1330A sodium
T69299
396731-20-7
AVE-1330A sodium is a beta-Lactamase inhibitor.
Antibacterial
Others
HIT214319341
Decaborane, diammonium salt
T31279
12046-71-8
Decaborane, diammonium salt is a biochemical.
Others
HIT214433610
Pelecopan
T62020
2378380-49-3
Pelecopan (BCX9930) 是有效的、选择性的口服补体因子D 抑制剂 (IC50= 14.3 nM)。Pelecopan 可以预防PNH 中的血管内和血管外溶血。
Complement System
Others
HIT105450635
N-BENZYL-2-PHENYLETHYLAMINE
T8629
3647-71-0
N-BENZYL-2-PHENYLETHYLAMINE 是 rel+ Escherichia coli B Phe-tRNA 的抑制剂。
Others
HIT214314689
PLGA
T19521
34346-01-5
PLGA (poly(lactic-co-glycolic acid)) 是一种聚乳酸和聚乙醇酸的共聚物,能够制造用于药物递送和组织工程应用的装置。
Others
HIT212031859
P7C3-A20
T2423
1235481-90-9
P7C3-A20 是促神经原性和神经保护活性的 P7C3 衍生物。它具有抗抑郁活性,能够透过血脑屏障,并可用于研究脑损伤。
Others
HIT212020074
4-Thiouridine
T35648
13957-31-8
4-Thiouridine (4-TU) 是一种光活化核糖核苷类似物,广泛用于RNA 分析。
Nucleoside Antimetabolite/Analog
Others
HIT103578963
Kipukasin D
T41107
948574-00-3
Kipukasin D is a naturally derived nucleoside with antibacterial properties, isolated from Aspergillus versicolor.
Antibacterial
Others
HIT212718379
T6A
T34765
24719-82-2
T6A (N6-Threonylcarbamoyladenosine) 是一种广泛存在具有普遍保守性的核苷,是修饰所必需的化合物。T6A 存在于负责转运 ANN 密码子的 tRNA 中。
Nucleoside Antimetabolite/Analog
Others
HIT214323805
Deoxythymidine-5'-triphosphate
T40467
365-08-2
Deoxythymidine-5'-triphosphate (dTTP) is a nucleoside triphosphate involved in DNA synthesis.
DNA/RNA Synthesis
Endogenous Metabolite
Nucleoside Antimetabolite/Analog
Others
HIT213334342
3'-Adenylic acid
T20055
84-21-9
3'-Adenylic acid 是一种生物活性化学剂。
cGAS
Nucleoside Antimetabolite/Analog
Others
HIT214435769
8-Methyl-2'-deoxyguanosine
TNU1523
85819-69-8
8-Methyl-2'-deoxyguanosine is a Nucleoside Derivative - 8-Modified purine nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214436038
5'-O-Benzoyl-2'-O,4'-C-methyleneuridine
TNU1577
293751-31-2
5'-O-Benzoyl-2'-O,4'-C-methyleneuridine is a Nucleoside Derivative - LNA related nucleoside; Protected nucleoside with NH2/OH open.
Nucleoside Antimetabolite/Analog
Others
HIT214436409
Tezacitabine
T60401
130306-02-4
Tezacitabine 是一种抑制细胞生长和细胞毒性的抗代谢物。 Tezacitabine 是一种核苷类似物,具有双重作用机制。 Tezacitabine 不可逆地抑制核糖核苷酸还原酶,并可在复制或修复过程中掺入 DNA,导致 DNA 链终止。 Tezacitabine 在细胞周期的 G1 期和 S 期阻断肿瘤细胞并诱导凋亡细胞死亡。 Tezacitabine 具有治疗白血病和实体瘤的潜力[1][2]。
Apoptosis
DNA/RNA Synthesis
Nucleoside Antimetabolite/Analog
Others
HIT214321586
Diadenosine pentaphosphate pentaammonium
T37309
102783-61-9
Diadenosine pentaphosphate pentaammonium, an endogenous vasoactive purine dinucleotide isolated from thrombocytes, is one component of the diadenosine polyphosphates (ApnA, n=2-7) family. These compounds are found in secretory vesicles, including those in platelets, chromaffin cells, Torpedo synaptic terminals, and brain synaptosomes[1][2].
Endogenous Metabolite
Others
HIT212666194
N6-Etheno 2'-deoxyadenosine
T19465
68498-25-9
N6-Etheno 2'-deoxyadenosine is used as a biomarker to evaluate chronic inflammation and lipid peroxidation in animal or human tissues.
Endogenous Metabolite
Nucleoside Antimetabolite/Analog
Others
HIT214433107
DMTr-LNA-C(Bz)-3-CED-phosphoramidite
TNU1570
206055-78-9
DMTr-LNA-C(Bz)-3-CED-phosphoramidite is a Nucleoside Phosphoramidite.
Nucleoside Antimetabolite/Analog
Others
HIT214433706
2'-O-Methyl-5'-O-dmt-inosine-3'-CE-phosphoramidite
TNU1561
128219-85-2
2'-O-Methyl-5'-O-dmt-inosine-3'-CE-phosphoramidite is a Nucleoside Phosphoramidite.
Nucleoside Antimetabolite/Analog
Others
Xanthine Oxidase
HIT214436267
2'-O-Acetyl-N4-benzoyl-5'-O-DMT arabinocytidine 3'-O-phosphoramidite
TNU1505
675573-97-4
Nucleoside Phosphoramidites;Arabino-nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT220912610
m7GpppUmpG
T74478
2638447-87-5
m7GpppUmpG,属于M7GpppNpG三核苷酸帽类似物的一种寡核苷酸,作为化学工具应用于具有cap 0或cap 1结构的RNA的合成。
Nucleoside Antimetabolite/Analog
Others
HIT214434740
3'-Azido-3'-deoxyguanosine
TNU0197
98870-11-2
Nucleoside Derivatives - Azido-nucleosides, 3'-Modified nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT214435771
2-Amino-6-chloro-9-(2-C-methyl-β-D-ribofuranosyl)-9H-purine
TNU0096
640725-74-2
2-Amino-6-chloro-9-(2-C-methyl-β-D-ribofuranosyl)-9H-purine is a 2'-C-Methyl nucleoside; Halo-nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT212044735
6-MPR
TNU0008
14675-48-0
6-MPR is a 2/6/8-modified purine nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214315140
IACS-8779
T11595
2243079-26-5
IACS-8779 is a potent STING agonist that efficiently stimulates interferon gene activity and exhibits strong systemic antitumor effects.
Others
STING
HIT214433744
2'-O-Hexadecanyl-2-aminoadenosine
TNU1653
2382942-28-9
2’-O-Hexadecanyl-2-aminoadenosine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU1653,CAS号为 2382942-28-9。
Nucleoside Antimetabolite/Analog
Others
HIT214432819
DMTr-TNA-U-amidite
TNU1608
325683-95-2
DMTr-TNA-U-amidite is a Nucleoside Phosphoramidite.
DNA/RNA Synthesis
Others
HIT214433657
3'-Azido-3'-deoxy-5-nitro-4-deoxyuridine
TNU0838
2072145-26-5
Nucleosides and Reagents - Azido-nuleoside; Pyridine nucleoside; 3'-N-Modified nucleoside
Nucleoside Antimetabolite/Analog
Others
HIT214432925
5'-O-(4,4'-Dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methyluridine
TNU1094
163759-50-0
5'-O-(4,4'-Dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methyluridine is a Nucleoside Derivative - 2'-Modified nucleoside; Protected nucleoside with NH2/OH open; Ready for further phosphorylation.
Nucleoside Antimetabolite/Analog
Others
HIT212033078
7-Deaza-2'-deoxy-7-iodoadenosine
T39141
166247-63-8
7-Deaza-2'-deoxy-7-iodoadenosine is a modified nucleotide containing 7-Deazaadenine.
DNA/RNA Synthesis
Others
HIT101719867
5'-Methylthioinosine
T125589
17298-58-7
5'-Methylthioinosine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125589,CAS号为 17298-58-7。
Others
HIT212028017
N6-Methyladenosine 5'-monophosphate disodium salt
T12162
81921-35-9
N6-Methyladenosine 5'-monophosphate disodium salt 是糖原磷酸化酶 b 激活剂,也是腺苷酸激酶 II 的抑制剂。
AChR
Others
Phosphorylase
HIT214435221
1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one
TNU0800
2072145-17-4
1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one is a Pyridine nucleoside; 2'-C-Methyl nucleoside.
Nucleoside Antimetabolite/Analog
Others
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