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2,4-Bipyridine是一种吡啶衍生物，广泛应用于生物化学实验和药物合成研究。

endogenous vanilloid TRPV1 (VR1) receptor agonist

Azide-PEG16-alcohol is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

DBCO-PEG4-Biotin (ADIBO-NH-PEG2-Biotin) 是一种 azadibenzocyclooctyne-biotin 衍生物，含有生物素基团和 4 个 PEG。DBCO-PEG4-Biotin 是一种用途广泛的生物素酰化试剂，能通过无铜催化烷基叠氮化反应 (SPAAC) 将生物素的一部分引入叠氮标记的生物分子中。

Boc-N-PEG5-C2-NHS ester is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Palmitoylisopropylamide 是一种选择性 FAAH 抑制剂，抑制[H]-AEA摄取，在低浓度下抑制细胞增殖。

2-Methylcyclopent-2-enone是一种环状酮，广泛应用于生物化学实验和药物合成研究。

PND-1186 hydrochloride (VS-4718 hydrochloride) 是高特异性的、可逆的 FAK 的有效抑制剂 (IC50: 1.5 nM)，能够选择性的诱导肿瘤细胞凋亡 (apoptosis)。

Regaloside C 是一种从百合属的中分离出来的甘油葡糖苷，具有抗炎作用。

Crotonyl-CoA，丁酸发酵、赖氨酸和色氨酸代谢中的关键中间体，对脂肪酸和氨基酸的代谢至关重要。

MW01-2-151SRM 是一种新型可穿过血脑屏障的小分子小胶质细胞活化抑制剂，具有抗神经炎作用，可减弱神经炎症模型中的神经胶质细胞因子上调，可用研究创伤性脑损伤、阿尔茨海默病和海藻氨酸毒性。

Isoastragaloside I 是一种中药黄芪的天然化合物，能够增强脂联素量活性。

(S, R, S)-AHPC-C8-NH2 (VH032-C8-NH2) is an E3 ligase ligand-linker conjugate. This compound comprises the VH032-based VHL ligand and a linker, specifically designed for AKT PROTAC degrader applications.

EM 5519 is an antitumor antibiotic.

Fructosyl-lysine (Fructoselysine) dihydrochloride 为通过美拉德反应由葡萄糖与赖氨酸反应生成的amadori glycation产物。该化合物是葡萄糖烷的前体，其中葡萄糖烷为一种赖氨酸-精氨酸蛋白交联物，常用作糖尿病检测的生物标志物。

'(R)-Preclamol hydrochloride ((+)-3-PPP hydrochloride)为Preclamol hydrochloride的R-对映异构体，作为DA激动剂，展现出对自身受体及突触后受体的刺激特性。'

PknB-IN-2 (Compound 10) 是一种结核分枝杆菌蛋白激酶B (PknB) 抑制剂 (IC50: 12.1 μM)。

16 alpha-Hydroxytrametenolic acid can inhibit 12-O-tetradecanoylphorbol 13-acetate (TAP)-induced mouse ear edema.

Hydroxy-PEG3-ethyl acetate is a polyethylene glycol (PEG)-based linker compound employed in PROTAC synthesis.

RM-018 is a powerful tricomplex inhibitor that specifically targets the active state of KRAS G12C. It exhibits unique functional characteristics and possesses the ability to bind and inhibit both KRAS G12C and KRAS G12C/Y96D, potentially overcoming resistance.

U-7524, also known as AOAA and Aminooxyacetic acid, is an inhibitor of 4-aminobutyrate aminotransferase (GABA-T). AOAA is also a general inhibitor of pyridoxal phosphate (PLP)-dependent enzymes (this includes GABA-T). It functions as an inhibitor by attac

Bumetanide sodium is a potent loop diuretic that acts as a blocker for the sodium-potassium-chloride cotransporter (NKCC). It selectively inhibits NKCC1 and NKCC2, with IC50 values of 0.68 μM and 4.0 μM for hNKCC1A and hNKCC2A, respectively [1] [2].

Cy5-PEG4-acid (chloride) serves as a PEG-based PROTAC linker, suitable for synthesizing PROTACs[1].

Hsp90-Cdc37-IN-1 is an Hsp90-Cdc37 interaction disruptor (IC50: 140 nM) that inhibit cell migration and reverse drug resistance.

Furosemide-d5是Furosemide的氘代标记物，可用于同位素示踪实验。Furosemide是 Na+/K+/2Cl- (NKCC)，NKCC1 和 NKCC2 共转运蛋白的有效的和具有口服活性抑制剂和GABAA 受体拮抗剂，用作利尿试剂、充血性心力衰竭，高血压和水肿的研究。

NSC16168 是一种选择性 ERCC1-XPF 抑制剂，可抑制 DNA 修复，增强顺铂的抗肿瘤活性。

CH2COOH-PEG6-CH2COOH is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

N-(Azide-PEG3)-N'-(PEG4-acid)-Cy5 is a PEG-based PROTAC linker employed for PROTACs (proteolysis-targeting chimeras) synthesis[1].

Cinchonain IIa has antioxidant activity, it shows high radical scavenging activity and reducing power.

Melflufen (Melphalan flufenamide) 是 Melphalan 的二肽前药，属于烷化剂。Melflufen 对多发性骨髓瘤（MM）细胞表现出显著的抗肿瘤活性，可抑制血管生成。Melflufen 能诱导 MM 细胞发生不可逆的 DNA 损伤和细胞毒性，发挥其抗肿瘤作用。Melflufen 的游离形式与盐形式表现出相似的生物活性。盐形式 Melflufen hydrochloride 通常具有更高的水溶性和稳定性。

Boc-PEG4-C2-NHS ester is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

DA 3003-2为一种高效的选择性Cdc25抑制剂，展示了抗增殖活性，能诱导细胞周期在G2/M期停滞，并提高P-tyr15Cdc2表达量，显示出对前列腺癌研究的应用潜力。

p38 MAPK-IN-2 is an inhibitor of p38 kinase.

Nevirapine (Standard) 是一种可用于分析的标准物质，通常用作 Nevirapine 的研究和分析中参考的标准样品。Nevirapine (NVP) 是一种 HIV-1逆转录酶非核苷抑制剂，Ki 值为 270 μM，可用于研究 HIV/AIDS。

Lithocholic acid 3-sulfate disodium (Standard) 是一种可用于分析的标准物质，通常用作 Lithocholic acid 3-sulfate disodium 的研究和分析中参考的标准样品。Lithocholic acid 3-sulfate disodium (Sulfolithocholic acid disodium) 可作为 RORgammat 配体，抑制 Th17 细胞分化。Lithocholic acid 3-sulfate disodium 是石胆酸（LCA）的硫酸化产物，可诱导细胞损伤。