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Laburnetin 是一种异黄酮类抗菌剂 (antibacterial agent)。Laburnetin 对真菌、S. vesicarium 具有抗菌活性。Laburnetin 增强了耐甲氧西林 (Methicillin) 金黄色葡萄球菌 (MRSA) 菌株对甲氧西林的敏感性。Laburnetin 可用于控制栽培物种的虫害。

Quorum sensing is a regulatory process used by bacteria for controlling gene expression in response to increasing cell density. This regulatory process manifests itself with a variety of phenotypes including biofilm formation and virulence factor production. Coordinated gene expression is achieved by the production, release, and detection of small diffusible signal molecules called autoinducers. The N-acylated homoserine lactones (AHLs) comprise one such class of autoinducers, each of which generally consists of a fatty acid coupled with homoserine lactone (HSL). AHLs vary in acyl group length (C4-C18), in the substitution of C3 (hydrogen, hydroxyl, or oxo group) and in the presence or absence of one or more carbon-carbon double bonds in the fatty acid chain. These differences confer signal specificity through the affinity of transcriptional regulators of the LuxR family. C14:1-δ9-cis-(L)-HSL is a long-chain AHL that functions as a signaling molecule in the quorum sensing of A. vitis. Regulating bacterial quorum sensing signaling can be used to inhibit pathogenesis and thus, represents a new approach to antimicrobial therpy in the treatment of infectious diseases.

Epirosmanol 是含有内酯部分的二萜类化合物。 Epirosmanol 是一种极弱碱性（基本中性）的化合物（基于其 pKa）。

4,5-Dimethyloxazole是一种噁唑类杂环化合物，广泛应用于生物化学实验和药物合成研究。

AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).

BPU-11 是一种 HCN4 CLP 配体，通过调节通道功能和完全消除 cAMP 诱导的 V1/2 变化来发挥作用。

ELOVL1-IN-1 (1-(2-Fluorophenyl)-N-(1-(2-fluoropyridin-4-YL)-1H-pyrazol-3-YL)cyclopropane-1-carboxamide) 是ELOVL1抑制剂，能够降低超长链脂肪酸的水平，可用于肾上腺脑白质营养不良的研究。

Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.

PDE4-IN-8 (Example 5) 是磷酸二酯酶4(PDE4)的有效抑制剂。PDE4-IN-8 对 PDE4B2 的 IC50值为 0.93 nM。然而，PDE4-IN-8 对 IL13、IL4、IFNy 的抑制作用微弱，IC50值分别为 4.04 nM, 36.33 nM, 2394 nM。

2-Ethylphenol (Standard)是一种可用于分析的标准物质，通常用作2-Ethylphenol的研究和分析中参考的标准样品。

6α-Hydroxy-5α-cholestane (6α-OHC) 是一种氧甾醇，可促进 SK-N-BE 细胞中超氧阴离子的产生。

Antibacterial agent 48 是一种抗菌剂，能够减少抗菌剂 Ceftazidime 的 MIC 值。

Tos-PEG4-t-butyl ester (Tos-PEG4-Boc) is a PROTAC linker characterized by its PEG composition. This compound plays a crucial role in the synthesis of a range of PROTACs, including BI-3663, a highly selective PTK2/FAK PROTAC. It employs cereblon ligands to target E3 ligases for the degradation of PTK2, exhibiting potent inhibitory activity with an IC50 of 18 nM[1].

BMS 310705 (21-Aminoepothilone B) 是 Epothilone B 的类似物，靶向卵巢癌、肾癌、膀胱癌和肺癌等恶性肿瘤。BMS 310705 通过线粒体介导的途径诱导显着的细胞凋亡 (apoptosis)。

Bis-NH2-C1-PEG3 (PROTAC Linker 24) is a polyethylene glycol (PEG)-based linker compound utilized in the synthesis of PROTACs. This compound serves as a critical component in constructing PROTAC molecules, facilitating the targeted degradation of specific proteins[1].

ICA-105665 (PF-04895162) 是一种有效的口服活性的神经元 Kv7.2/7.3和 Kv7.3/7.5钾通道激动剂。ICA-105665 在人肝细胞中具有低细胞毒性潜力，但抑制肝线粒体功能和胆盐输出蛋白 (BSEP) 转运 (IC50为 311 μM)。ICA-105665 可穿透中枢神经系统 (CNS)并具有抗癫痫作用。

NSC114126 is a highly effective and orally bioavailable inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor (EGFR-TK). This compound exhibits robust antiproliferative properties, making it a promising candidate for further investigation in the field of cancer research [1].

AZD1092 is the glucokinase enzyme activator.

tachykinin NK1 receptor antagonist

Neopentylamine是一种伯胺，广泛应用于生物化学实验和药物合成研究。

2-(3-methyl-1H-1,2,4-triazol-5-yl)aniline是一种高纯度生化试剂，可作为特异性探针辅助解析含氮杂环化合物的生化作用机制用于生物化学实验和药物合成研究。

DNP-PEG4-alcohol is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Inz-4 is a fungal-selective inhibitor of mitochondrial cytochrome bc1.

Methyltetrazine-PEG8-NHS ester is a polyethylene glycol (PEG) derivative, specifically designed as a PROTAC linker for the synthesis of Proteolysis Targeting Chimeras (PROTACs)[1].

Prothipendyl hydrochloride 适用于研究老年人精神症状（例如焦虑）。

Remikiren is a highly specific renin inhibitor with oral activity for the treatment of hypertensio.

CGP78850 is a potent and selective Grb2 SH2-phosphopeptide interaction antagonist that holds potential for cancer research.

Difluprednate (Myser) 是一种可用于术后眼睛疼痛和炎症的皮质类固醇。

GNE-4997 is a potent and selective inhibitor of the interleukin-2-inducible T-cell kinase (Ki: 0.09 nM). The correlation between the basicity of solubilizing elements in GNE-4997 and off-target antiproliferative effects decreases cytotoxicity.

CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.

Ladostigil hemitartrate (TV-3326) is a compound that acts as a dual inhibitor of cholinesterase and brain-selective monoamine oxidase (MAO). It has IC50 values of 37.1 μM for MAO-B and 31.8 μM for AChE. In addition, Ladostigil hemitartrate possesses neuroprotective, antioxidant, and anti-inflammatory properties. It is commonly used in research relating to depression and Alzheimer's disease.

AKV-9 是一种突变型 Cu/Zn 超氧化物歧化酶（SOD1）抑制剂，能够有效抑制 SOD1 诱导的蛋白聚集，并在 PC-12 细胞中对抗 SOD1 诱导的细胞毒性，EC50 为 0.3 μM。AKV-9 还能改善肌萎缩侧索硬化症（ALS）相关表型并显著延长小鼠模型的生存期，适用于 ALS 发病机制及靶向治疗研究。

Tuberculosis inhibitor 12（compound 12）作为恶二唑衍生物，表现出对结核分枝杆菌的显著抑制作用。在7H9-Tw-OADC介质中，Tuberculosis inhibitor 12（20 μM）展现了82%的抑制率，而在相同条件下抑制率为78%。

Dipyrithione 似乎具有新的细胞毒性和强大的广谱抗肿瘤活性。

Zaurategrast ethyl ester is the ethyl ester prodrug of CT7758 and is an α4β1/α4β7 integrin antagonist. It is used for the treatment of inflammatory and autoimmune disorders.

Tarazepide is a potent and specific antagonist of CCK-A receptor.