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供应商货号
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HIT ID
供应商货号
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Others
Advanced Glycation End Products
CYP19A1
Decarboxylase
DprE1
Fer/FerT kinase
Platelet aggregation
Progesterone Receptor
Others
信号通路
其他
Others
Others
Targetmol为生命科学及医药领域的科研人员提供其他未细分细胞信号通路相关产品,包括抑制剂、激动剂、调节剂、降解剂等。
HIT217590805
2-MT-63
T68484
870225-11-9
2-MT 63 is a novel TIE-2 kinase inhibitor that demonstrates unique and improved kinase selectivity compared to other inhibitors known to interact with TIE-2. 2-MT 63 has a good kinase selectivity profile in enzyme assays with >30-fold selectivity (typically much greater) against the tested kinases. Importantly, the profile includes selectivity against other targets of relevance for angiogenesis (KDR, PDGFR, EPHB4).
Others
Tie-2
HIT214982325
Desvaleryl Valsartan
T68890
676129-92-3
Desvaleryl valsartan is a potential impurity found in commercial preparations of the angiotensin II type 1 (AT1) receptor antagonist valsartan. It is a degradation product formed under acidic conditions.
Drug Metabolite
Others
HIT215320306
OL-135
T68881
681135-77-3
OL-135 is a CNS penetrant, highly potent and selective reversible inhibitor of FAAH. OL-135 exhibits analgesic pharmacology in various animal models without the motor impairment associated with direct CB1 agonism.
FAAH
Others
HIT215476390
KU-0058684
T68978
623578-11-0
KU-0058684 is a potent PARP and DNA-PK inhibitors.
Others
PARP
HIT212078982
Clozapine HCl
T69129
54241-01-9
Clozapine HCl is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays a unique pharmacological profile. Clozapine is a serotonin antagonist, with strong binding to 5-HT 2A/2C receptor subtype. It also displays strong affinity to several dopaminergic receptors, but shows only weak antagonism at the dopamine D2 receptor, a receptor commonly thought to modulate neuroleptic activity. Agranulocytosis is a major adverse effect associated with administration of this agent.
5-HT Receptor
AChR
Adrenergic Receptor
Dopamine Receptor
Others
HIT213886176
Harmol hydrochloride monohydrate
TN4184
40580-83-4
Harmol hydrochloride monohydrate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4184,CAS号为 40580-83-4。
Monoamine Oxidase
Others
HIT214316951
12-Deoxo-12α-acetoxyelliptone
TN5452
150226-21-4
12-Deoxo-12alpha-acetoxyelliptone is a natural product from Derris robusta.
Others
HIT213885744
Oleuropeic acid 8-O-glucoside
TN4706
865887-46-3
Oleuropeic acid 8-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4706,CAS号为 865887-46-3。
Antibacterial
Others
HIT213884502
14-Deoxy-17-hydroxyandrographolide
TN2623
869384-82-7
14-Deoxy-17-hydroxyandrographolide是一种天然产物,属于爵床科穿心莲属,其产品编号为 TN2623,CAS号为 869384-82-7。14-Deoxy-17-hydroxyandrographolide可用作对照参考。
Antifection
Others
HIT214435885
2-Methoxy-2'-deoxy-2'-fluoro-beta-D-arabinoadenosine
TNU0081
1093278-52-4
Fluoro-modified nucleoside; 2/6/8-Modified purine nucleoside; Arabino-nucleoside
Nucleoside Antimetabolite/Analog
Others
HIT214435771
2-Amino-6-chloro-9-(2-C-methyl-β-D-ribofuranosyl)-9H-purine
TNU0096
640725-74-2
2-Amino-6-chloro-9-(2-C-methyl-β-D-ribofuranosyl)-9H-purine is a 2'-C-Methyl nucleoside; Halo-nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT212044735
6-MPR
TNU0008
14675-48-0
6-MPR is a 2/6/8-modified purine nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214433522
5-Iodo-3'-deoxy-3'-fluorouridine
TNU0013
2072145-21-0
5-Iodo-3'-deoxy-3'-fluorouridine is a Nucleoside, fluoro-modified nucleoside, halo-nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214433198
Arabinoisocytidine
TNU0051
10212-30-3
Isocytidine derivative; Arabino-nucleoside
Nucleoside Antimetabolite/Analog
Others
HIT212020591
4'-alpha-Azidouridine
TNU0015
139442-01-6
4'-alpha-Azidouridine is a Nucleoside-Azido-nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214436421
6-(Furan-2-yl)purine-beta-D-(3'-deoxy-3'-fluoro)riboside
TNU0017
1612191-89-5
Nucleoside Derivatives - Fluoro-modified nucleosides; 6-Modified purine nucleosides, 3'-Modified nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT214434571
5-Iodo-2'-O-methylcytidine
TNU0018
847650-69-5
5-Iodo-2'-O-methylcytidine is a Halo-nucleoside; 2'-O-Methyl nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214435490
5-(Trifluoromethyl)uridine
TNU0032
21618-67-7
5-(Trifluoromethyl)uridine is a Nucleoside Derivative - Fluoro-modified nucleoside, 5-Modified pyrimidine nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214435866
2'-Chloro-2'-deoxycytidine
TNU0074
10212-19-8
Nucleoside Derivatives - Halo-nucleosides, 2'-Modified nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT214432931
6-Methylpseudouridine
TNU0076
1613530-10-1
6-Methylpseudouridine is a Nucleoside Derivative - C-nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214435716
2-Amino-2′-C-methyladenosine
TNU0110
640725-73-1
2-Amino-2'-C-methyladenosine is a 2'-C-Methyl nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214434215
2-Chloro-2'-C-methyl-6-N,N-dimethyladenosine
TNU0111
2095417-43-7
2'-C-Methyl nucleoside; Halo-nucleoside; 2/6/8-Modified purine nucleoside
Nucleoside Antimetabolite/Analog
Others
HIT214433252
2'-C-b-Methyl-4-deoyuridine
TNU0114
1106032-88-5
Nucleosides and Reagents - 4-Deoxypyrimidine nucleoside; 2'-C-Methyl nucleoside
Nucleoside Antimetabolite/Analog
Others
HIT214434700
5-Pyrrolidinomethyluridine
TNU0121
1613530-41-8
5-Pyrrolidinomethyluridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Scaffold and Template.
Nucleoside Antimetabolite/Analog
Others
HIT214436381
5-(N-Isopentenyl-N-trifluoroacetyl) aminomethyluridine
TNU0120
1613530-43-0
5-(N-Isopentenyl-N-trifluoroacetyl) aminomethyluridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Amino nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214435272
N1-Benzyl pseudouridine
TNU0117
1613530-22-5
N1-Benzyl pseudouridine is a Nucleoside Derivative - C-nucleoside; N-Methylated nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214436118
2'-C-Methyl-2-thiouridine
TNU0135
1678507-60-2
2'-C-Methyl-2-thiouridine is a Nucleoside Derivative - Thio-nucleoside, 2'-Modified nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214433084
1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine
TNU0385
2389988-20-7
1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside; Amino nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214433761
N4,N4-Dimethylarabinocytidine
TNU0392
82855-64-9
N4,N4-Dimethylarabinocytidine is a Nucleoside Derivative - Arabino-nucleoside, N-Methylated nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214435824
N4-Methylarabinocytidine
TNU0391
13491-42-4
N4-Methylarabinocytidine is a Nucleoside Derivative - Arabino-nucleoside, N-Methylated nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214435296
1-Amino-7-cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl)guanine
TNU0387
2389988-22-9
Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; Amino nucleosides; N-Methylated alkylated nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT214436201
1-(b-D-Xylofuranosyl)-2-thiouracil
TNU0371
2305416-17-3
Nucleoside Derivatives - Xylo-nucleosides, Thio-nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT214435977
8-Allyloxyadenosine
TNU0364
2095417-69-7
8-Allyloxyadenosine is a Nucleoside Derivative - 8-Modified purine nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214434047
N3-Methyl-2'-O-(2-methoxyethyl)uridine
TNU0375
2305416-12-8
N3-Methyl-2'-O-(2-methoxyethyl)uridine is a Nucleoside Derivative - N-Methylated nucleoside.
Nucleoside Antimetabolite/Analog
Others
HIT214436173
2',3'-Anhydro-tubercidin
TNU0416
40627-31-4
Nucleoside Derivatives - 7-Deaza-purine nucleosides; Anhydro-nucleosides
Nucleoside Antimetabolite/Analog
Others
HIT214434455
3'-Deoxy-3'-fluoro-5-trifluoromethyluridine
TNU0141
439579-21-2
3'-Deoxy-3'-fluoro-5-trifluoromethyluridine is a nucleoside and Reagent - Fluoro-modified nucleoside; 5-Modified pyrimidine nucleoside.
Nucleoside Antimetabolite/Analog
Others
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