Others

NC1153 is a blocker of IL-2-induced activation of JAK3 and its downstream substrates STAT5a/b. It promotes long-term allograft survival and sparing the recipient from multiple toxicities.

Mirincamycin HCl is a close analog of the drug clindamycin used for the treatment of Plasmodium falciparum blood stages.

N-Acetylpurinomycin is a selective agonist of CB2 receptor.

Nopol is an inhibitor of alpha-glucosidase.

Aviglycine is an antibiotic.

Diallyl G is a delta-opioid receptor antagonist agent.

Dipiproverine 是α-氨基酸酯类化合物，是一种解痉化合物。它被用作抗胆碱能药物。

Detoxin C1 is a selective blasticidin S antagonist.

Cyanopeptolin 954 is a chlorine-containing Microcystis aeruginosa NIVA Cya 43 chymotrypsin Inhibitor.

Ecraprost is used as a prodrug of prostaglandin E1.

LEK 8841 is an ergoline derivative that is a potential antipsychotic.

Folitixorin calcium is an antineoplastic enhancing agent.

Levamlodipine gentisate is a pharmacologically active enantiomer of amlodipine. Amlodipine is the dihydropyridine calcium channel blocker used as an antihypertensive and antianginal drug.

LDN-193665 is a potent inhibitor of tau kinase. It acts by targeting CDK5​/p25 and GSK3β.

Fenclofenac is a non-steroidal anti-inflammatory agent that competitively supresses the binding of thyroxine(T4) and triiodothyronine (T3) by thyroxine-binding globulin(TBG).

TAS-4 is a modulator of metabotropic glutamate receptor 4-positive allosteric.

L 738372 is a non-nucleoside inhibitor of HIV-1 reverse transcriptase.

L 722151 is an FXIIIa inhibitor.

AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.

L 158809 is an antagonist of the angiotensin II type 1 receptor.

Men 10208 is an antagonist of the neurokinin A receptor.

NS4591 is a modulator of SK-IK channels.

Anirolac is a nonsteroidal anti-inflammatory agent.

Vif-A3G Inhibitor N.41 is a HIV-1 inhibitor-targeting drug. It causes Vif-dependent degradation of human APOBEC3G, thereby inhibiting the Vif-A3G interaction.

Seriniquinone is a selective agent of anticancer that acts by inducing cell death via autophagocytosis and targeting the cancer-protective protein dermcidin.

H-0104 Dihydrochloride is an inhibitor of ROCK that acts by applying potent intraocular pressure (IOP)-lowering effects into the eyes of monkeys.

Prumycin is an agent of antifungal antibiotic.

CFM-1 is an antagonist of the anaphase-promoting complex (APC)-2. It also is a cell cycle and apoptosis regulatory protein (CARP)-1 interaction antagonist.

H2-005 is a selective inhibitor of diacylglycerol acyltransferase 2 (DGAT2).

L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.

L 659989 is an antagonist of the Platelet-activating factor receptor.

Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.

Letimide HCl is an analgesic agent.

Lanceotoxin A is a potent Ip blocker.

Linearol is a diterpene found in Sideritis L. spp. (Lamiaceae) with a broad range of demonstrated properties including antioxidant, anti-inflammatory, and anti-apoptotic activities.

Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.