Others

7ETMC is a selective Human Cytochrome P450s 1A1 and 1A2 inhibitor. 7ETMC showed IC50s of 0.46 μM and 0.50 μM for P450s 1A1 and 1A2 in the first six minutes, respectively, and did not show any inhibition activity for P450s 2A6 and 2B1 even at the dose of 5

Lincophenicol is an Escherichia coli ribosomal peptidyltransferase-catalyzed puromycin reaction inhibitor.

LY 173013 is a bicyclic pyrazolidinone, it has antibacterial properties.

MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.

ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.

KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.

OMDM169 is a potent and selective MAGL inhibitor. OMDM169 could enhances 2-AG levels and of exerts analgesic activity via indirect activation of cannabinoid receptors. OMDM169 exhibited 0.13 microM<IC(50)<0.41 microM towards 2-AG hydrolysing activities in

Ono-3805 is an inhibitor of nonsteroidal 5 alpha-reductase.

GSK926 is a selective, SAM-competitive, and cell-active EZH2 inhibitor.

Bisaramil is a new class I antiarrhythmic agent.

Griselimycin is a natural antimycobacterial product that is currently being pursued as a therapy for tuberculosis.

BMS 180742 is an exosite inhibitor of thrombin.

Hexadecylphosphoserine is a representative growth inhibitor.

Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.

Bifidenone is an effective tubulin polymerization inhibitor.

Benmoxin is a monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective.

MDK-4683, also known as CA IX/XII Inhibitor, is a hCA IX and hCA XII inhibitor.

Pentamethonium bromide is a vasodilator agent.

Phox-I1 is a NOX2 inhibitor targeting the interactive site of p67phox with Rac GTPase.

NU/ICRF 500 is a novel anthracenyl-amino acid catalytic inhibitor of topoisomerase II.

NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.

Razobazam is a benzodiazepine derivative agent. It produces nootropic (improves cognitive function) effects in animal studies.

Rev 6207 is a non-sulfhydryl ACE-inhibitor.

S-Aristeromycinylhomocysteine is an inhibitor of adenosylmethionine decarboxylase.

JY-XHe-053 is a selective modulator of GABAA receptors.

KKJ00626, an inhibitor of HBV virus, inhibits HBV replication in transfected Huh7 cells.

MRS1067 is an antagonist of A3 adenosine receptor.

LSP1-2111 is a mGlu4 receptor subtype agonist.

Lombazole is an antimicrobial agent in the class of imidazole.

LY 215490 is a selective, competitive and systemically active antagonist of AMPA receptor. LY 215490 has neuroprotective effect against focal ischaemia in a model of permanent MCA occlusion in the rat.

LTURM-36 is a novel inhibitor of PI 3-kinase delta.

MRT-68601 HCl, a potent TBK1 (TANK-binding kinase-1), inhibits the formation of autophagosomes in lung cancer cells.

FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.

DW10075, a novel potent and highly selective inhibitor of VEGFR, exhibits antitumor activities both in vitro and in vivo.

Guanoctine hydrochloride has antihypertensive activity.

Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.