Others

Ripazepam has anxiolytic effects.

Chitin synthase inhibitor 3 (compound 2d) 是一种高效的chitin synthase抑制剂，具有0.16 mM的IC50值，并对candida albicans显示出1 μg/mL的MIC，表现出抗真菌活性。

Adenosine receptor antagonist 3 具有用于癌症疾病研究的潜力，它是腺苷受体的有效拮抗剂。

Squalamine lactate is an aminosterol compound discovered in the tissues of the dogfish shark, with antimicrobial activity.

2,3-Heptanedione（2,3-庚烷二酮）是一种酮，常用于香料制备、有机合成和生化实验。

Epothilone E，作为Epothilone的衍生化合物，通过抑制微管蛋白功能来阻碍细胞分裂，从而展现出抗肿瘤活性。

m-PEG10-Tos is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Boc-NH-PEG3-propargyl is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

FTO-IN-5 是一种有效且选择性的脂肪量和肥胖相关蛋白（FTO）抑制剂。

(S)-1-(4-Hydroxyphenyl)ethane-1,2-diol 是当归地上部分的主要活性成分，能显著抑制嗜水气单胞菌的生长，并具有抗凝及抗生素活性。

N-Desmethylnefopam is the main Nefopam metabolite .

Micafungin sodium (Standard) 是一种可用于分析的标准物质，通常用作 Micafungin sodium 的研究和分析中参考的标准样品。Micafungin sodium (FK 463) 是抗真菌剂，抑制1, 3-beta-D-glucan 的合成。

1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid (Nudifloric Acid) 是来源于冬虫夏草，能够靶向阻断 AP-1 介导的荧光素酶活性，具有抗炎活性。其中冬虫夏草具有抗氧化，抗癌，抗炎，抗糖尿病，抗肥胖，抗血管生成和抗伤害感受活动。

Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.

DS86760016 is a highly effective inhibitor of leucyl-tRNA synthetase (LeuRS), demonstrating potent activity against multidrug-resistant (MDR) Gram-negative bacteria including Escherichia coli, Klebsiella pneumoniae, and Pseudomonas aeruginosa. Notably, DS86760016 effectively inhibits LeuRS enzymes derived from Escherichia coli, Pseudomonas aeruginosa, and Acinetobacter baumannii, exhibiting IC50 values of 0.38 μM, 0.62 μM, and 0.16 μM, respectively.

Okilactomycin is a biochemical.

Prifinium bromide是抗胆碱能试剂，能够改善痉挛，具有止吐效果。

Uzansertib (INCB053914) is a potent ATP-competitive pan-PIM kinase inhibitor. It exhibits exceptional inhibitory activity against PIM1, PIM2, and PIM3 with IC50 values of 0.24 nM, 30 nM, and 0.12 nM, respectively. Furthermore, Uzansertib demonstrates significant anti-proliferative effects against an assorted range of hematologic tumor cell lines.

Namoline is a γ-pyrone compound that functions as a selective and reversible inhibitor of Lysine-specific demethylase 1 (LSD1) with an IC50 of 51 μM in an HRP-coupled enzymatic assay. By impairing LSD1 demethylase activity, Namoline effectively inhibits cell proliferation. Due to its characteristics, Namoline holds promise for research pertaining to androgen-dependent prostate cancer.

Tripotassium citrate是一种含有钾离子的柠檬酸，在生化实验中常用于缓冲剂，在有效范围内保持稳定的pH值。Tripotassium citrate也可用于治疗尿路结石。

CDK12-IN-6, a pyrazolotriazine compound, is a powerful inhibitor of CDK12. Its inhibitory activity is significant with an IC50 value of 1.19 μM when tested at high ATP concentration (2 mM). Notably, CDK12-IN-6 does not exhibit any inhibitory effect on CDK2/Cyclin E (IC50 >20 μM) and CDK9/Cyclin T1 (IC50 >20 μM) when tested under the same high ATP conditions (2 mM) (WO2021116178A1).

Corydamine 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T124768。

Bis-sulfone-PEG4-DBCO is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Estramustine phosphate can be used to treat prostatic neoplasms; also has radiation protective properties.

B-Raf IN 8 (compound 7g) 是 B-Raf 的有效抑制剂 (IC50 = 70.65 nM)。B-Raf IN 8 显示出抗肿瘤活性，其对肝细胞癌 (HEPG-2)、结肠癌 (HCT-116)，乳腺癌 (MCF-7) 和人前列腺癌 (PC-3) 细胞的 IC50值分别为9.78、13.78、18.52 和 29.85 μM。

Omeprazole magnesium 是口服活性的质子泵（proton pump）抑制剂（PPI），用于抑制胃酸，常用于研究胃酸反流和烧心症相关症状。

Fmoc-PEG24-NHS ester is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Clofazimine (Standard) 是一种可用于分析的标准物质，通常用作 Clofazimine 的研究和分析中参考的标准样品。Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料，与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。

1-Penten-3-ol是一种含有双键和羟基的有机化合物，广泛应用于生物化学实验和药物合成研究。

LUF7346 is an allosteric modulator of hERG.

sEH/AChE-IN-3 -15) 是一种有效的、可透过血脑屏障的 sEH(可溶性环氧水解酶)和 AChE(乙酰胆碱酯酶)的双重抑制剂，其 IC50分别为 0.4 nM (hsEH)、1.94 nM (hAChE)、615 (hBChE，丁酰胆碱酯酶)、4.3 nM (msEH) 和 2.61 nM (mAChE)。

iGP-1 是一种线粒体sn-甘油3-磷酸脱氢酶（mGPDH）抑制剂，可用于研究肥胖。

2,7-Dimethylnaphthalene是一种多环芳烃（PAH）衍生物，广泛应用于生物化学实验和药物合成研究。

8-Hydroxyadenosine (8-Oxoadenosine) 是一种存在于 Torula 酵母 RNA 中的嘌呤核苷。

Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) 是一种有效的选择性 N-甲基-D-天冬氨酸受体激动剂。

BRD7552 是PDX1转录因子诱导剂，它能够上调人类原代胰岛和导管细胞中 PDX1 的表达，诱导 PDX1 启动子的表观遗传变化与转录激活一致，提高胰岛素表达。其中 PDX1 是参与胰腺发育和β细胞功能的关键转录因子。