Others

Bioresmethrin is a pesticide of synthetic pyrethroid.

TNIR7-1A 是一种环庚三烯-BODIPY 衍生物，具有适用于近红外 (NIR) 成像的特性（PBS 中的 Ex/Em = 600/774 nm），并且在体外对神经原纤维缠结 (NFT) 展现出高亲和力和特异性。同时，TNIR7-1A 能够有效穿透血脑屏障。

Enpp-1-IN-21 (compound 4g) 是一种外核苷酸焦磷酸酶/磷酸二酯酶 1 (ENPP1) 的抑制剂，其对ENPP1和ENPP3的IC50分别为0.45 μM和0.19 μM。

I194496，一种有效的cystathionine γ-lyase (CSE)抑制剂，其IC50值达到0.79 mM。该化合物不仅能通过双重靶点PI3K/Akt和Ras/Raf/ERK通路抑制人类TNBC细胞的生长，还可以通过下调Anxa2/STAT3和VEGF/FAK/Paxillin信号通路，进一步抑制人类TNBC细胞的转移。

Iodoacetic anhydride是具有酶活性抑制特性的生物活性化合物。该化合物能够参与蛋白质修饰，因此广泛用于生物化学研究和化合物开发。此外，Iodoacetic anhydride也被用于合成多种生物活性分子，展现了其作为化学试剂的广泛应用性。

Row174336 (compound 29) 作为Hsp110-STAT3相互作用的有效抑制剂，显示出对HPAEC细胞系的抗增殖效果，其IC50值为22.67 μM。

Nostopeptin B is an inhibitor of elastase.

J1075 is an histone deacetylase 8 (HDAC8) inhibitor.

Miloxacin is an antibiotic active against gram-negative bacteria.

Levonadifloxacin, a broad-spectrum fluoroquinolone antibiotic, is used potentially for the treatment of staphylococci.

LY 221068 is a potent antioxidant with anti-inflammatory activity.

M199, a novel inhibitor of TLR3/9 activation, induces secretion of IL-6, IL-8 and TNFalpha in human PBMCs.

Camylofin HCl is an antispasmodic used in labor treatment and is also used to deliver drug therapy for ulcerative colinitis.

Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.

Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.

PIK-C98 is an inhibitor of PI3K that acts by displaying potent preclinical activity against multiple myeloma.

546C88 is an inhibitor of nitric oxide synthase.

Antibiotic K 4 is an inhibitor of angiotensin I converting enzyme produced by Actinomadura spiculosospora.

(E/Z)-LAQ824 is an inhibitor of histone deacetylase.

E-982 is derived from the reference compound.

Solabegron (GW-427,353), is a selective agonist of β3 adrenergic receptors. In addition, Solabegron has been shown to produce visceral analgesia by releasing somatostatin from fat cells.

Vapreotide diacetate is a synthetic analog of somatostatin. It has analgesic activity most likely mediated through the blockade of the neurokinin-1 receptor (NK1R), the substance P (SP)-preferring receptor.

3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.

BN 50341 is an inhibitor of antithrombotic platelet activating factor.

ADX-10061 is a dopamine D1 receptor antagonist.

A-176120 is a potent farnesyl pyrophosphate (FPP) analogues, it selectively inhibits farnesyltransferase. It has anti-angiogenic potential and may reduce H-ras NIH3T3 tumour growth.

CM-414 is a dual inhibitor of HDACs and PDE5 for the Treatment of Alzheimer’s Disease (IC50 values of 60 nM, 310 nM, 490 nM, 322 nM, and 91 nM against PDE5, HDAC1, HDAC2, HDAC3, and HDAC6, respectively). Chronic treatment of Tg2576 mice with CM-414 dimini

Tylophorine analog DCB-3503 is a potential anticancer and immunosuppressive agent. DCB-3503 suppresses the translation of cellular regulatory proteins, including cyclin D1, at the elongation step. DCB-3503 allosterically regulates the ATPase and chaperone activities of HSC70 by promoting ATP hydrolysis in the presence of specific RNA binding motifs (AUUUA) of cyclin D1 mRNA.

R 115777 is an inhibitor of farnesyl transferase.

Rooperol is a norlignan derivative with numerous biological activities including immunomodulatory, antitumor, antibacterial, anticonvulsant, and antioxidant activities. It is a novel p38α inhibitor.

SK&F 104976 is a 32-carboxylic acid derivative of lanosterol. It was found to be a potent lanosterol 14 alpha-demethylase (14 alpha DM) inhibitor.

ABD56 inhibits osteoclast formation and activity in vitro and in vivo.

BO 1165 is an monobactam antibiotic.

Cameglipti, a dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type 2 diabetes.

MHY884 is an inhibitor of tyrosinase that acts by inhibiting UVB-induced activation of the NF-κB signaling pathway through the downregulation of oxidative stress.

DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.