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Benzyl-PEG4-MS 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T67180，CAS号为 477781-69-4。

Bendazac (Bendazolic acid) 是一种氧乙酸，具有抗过敏、抗炎、利胆和抗血脂作用。它能够阻断蛋白质变性，延缓白内障的发生过程。

SCH 51344 抑制Ras 诱导的恶性转化。SCH 51344可防止癌基因转化的成纤维细胞的非锚定生长。

Valopicitabine, a NS5B inhibitor, is used potentially for the treatment of HCV infection.

ACT-209905 is an agonist of S1P1 receptor.

AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM).

1,16-Hexadecanediol 毒性较低，可用于制作树脂和纳米材料。

AZ8838 是一种有效的、竞争性的、变构的、口服活性的 PAR2非肽小分子拮抗剂，其对 hPAR2 的 pKi 值为 6.4。

Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.

MrgprX2 antagonist-4 and compound B-51 E117, is a potent MrgprX2 antagonist. It specifically targets and inhibits the MrgprX2 receptor, making it suitable for investigating various inflammatory skin disorders.

Clofibrin is a kind of hypolipidemic drug, which can reduce Hypertriglyceride and hypercholesterolemia.

FR 901465 is a biochemical.

BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).

Axl-IN-9 是一种 AXL 的有效抑制剂 (IC50: 26 nM)，具有优良的跨膜性。Axl-IN-9 在动物体内表现出良好的药代动力学特性。Axl-IN-9 能够用于研究增生性疾病、自身免疫性疾病、过敏性疾病、移植排斥、炎症性疾病、癌症或其他哺乳动物疾病。

(R)-Necrocide 1（化合物(R)-38）是一种具有抗增殖活性的有效抗癌剂。

2',4',6'-trihydroxy-3'-(3-methyl-2-butenyl)acetophenone是一种天然的苯乙酮衍生物，可用于生物化学实验和药物合成研究。

Pseudoneolinderane是一种发现于Neolitsea aciculata Koidz的倍半萜烯，可用于生物化学实验和药物合成研究。

Orexin 2 Receptor Agonist 2 (ORA-2) is a specific agonist for the orexin 2 receptor.

S-acetyl-PEG4-NHBoc is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

HDAC-IN-31 是一种选择性的、有效的、口服具有活力的 HDAC 抑制剂，能够作用于 HDAC1 (IC50: 84.90 nM)、HDAC2 (IC50: 168.0 nM)、HDAC3 (IC50: 442.7 nM)、HDAC8 (IC50>10000 nM)。 HDAC-IN-31 能够将细胞周期阻滞在 G2/M 期，并诱导细胞凋亡 (apoptosis)。HDAC-IN-31 具有良好的抗肿瘤效果。HDAC-IN-31 对弥漫性大 B 细胞淋巴瘤表现出潜在的研究价值。

TP-050 是一种口服有效的选择性 NMDAR 激动剂，抑制 GluN2A 和 GluN2D 的 EC50值分别为 0.51 μM 和 9.6 µM。TP-050 可穿过血脑屏障 (BBB)。TP-050 诱导海马区的长期增益效应 (LTP)，增强神经元信号传输。

AMG 487 is an effective and selective antagonist of chemokine receptor 3. AMG 487 inhibited CXCR3-mediated cell migration induced by three CXCR3 chemokines, IP-10, ITAC and MIG (IC50: 8, 15 and 36 nM, respectively).

m-PEG5-phosphonic acid is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Thalidomide-O-C6-NH2 TFA is a synthesized E3 ligase ligand-linker conjugate used in the PROTAC dTAG-13, a degrader of FKBP12F36V and BET[1].

DNP-PEG4-DBCO is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

HS-PEG5-CH2CH2N3 is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

Guanadrel 是一种抗高血压药。

ATR-IN-16 (compound 46) is a highly effective ATR kinase inhibitor, exhibiting considerable anticancer activity in LoVo cells, as demonstrated by its IC 50 value of 410 nM [1].

HA15-Biotin is a chemically synthesized compound comprising HA15 which is connected to biotin through the amide group. It demonstrates comparable activity to HA15 and holds potential for use in proteomic analysis.

Empagliflozin (Standard) 是一种可用于分析的标准物质，通常用作 Empagliflozin 的研究和分析中参考的标准样品。Empagliflozin (BI 10773) 是一种 SGLT-2 抑制剂 (IC50=3.1 nM)，具有有效的和选择性，对 SGLT-1/4/5/6 的选择性高 300 倍以上。Empagliflozin 可用于治疗二型糖尿病。

Regorafénib N-oxyde (M2) (Standard) 是一种可用于分析的标准物质，通常用作 Regorafénib N-oxyde (M2) 的研究和分析中参考的标准样品。Regorafénib N-oxyde M2 是 Regorafenib 的活性代谢物。Regorafenib 是多靶点抑制剂，包括VEGFR1/2/3，PDGFRβ，Kit，RET 和 Raf-1 ， IC50分别是 13/4.2/46，22，7，1.5 和 2.5 nM。

Antibacterial agent 116 是一种含二苯甲酮的水杨酰苯胺类化合物。Antibacterial agent 116 能抑制肽聚糖的形成而具有较强的抗菌活性。Antibacterial agent 116 可作为光亲和探针标记 Acinetobacter baumannii 的青霉素结合蛋白 (PBP1b)，干扰肽聚糖链的生长，阻断其增殖。

IDO1-IN-18 (Compound 14) 是一种 IDO1 的有效抑制剂。IDO1-IN-18 具有潜力进行癌症疾病的研究。

GGTI-2154 hydrochloride 是一种有效的、选择性的 geranylgeranyltransferase I (GGTase I) 抑制剂 (IC50: 21 nM)。GGTI-2154 hydrochloride 对 GGTase I 的选择性是 FTase (IC50: 5600 nM) 的 200 倍以上。GGTI-2154 hydrochloride 能够用于研究癌症。

Gliclazide is a whole-cell beta-cell ATP-sensitive potassium currents blocker with an IC50 of 184 nM. Ethyl tosylcarbamate is an intermediate in the synthesis of Gliclazide (G409877).

Propargyl-PEG3-amine is a PEG derivative containing a propargyl group and an amino group. The propargyl group can be reacted with azide-bearing compounds or biomolecules via copper-catalyzed azide-alkyne Click Chemistry to yield a stable triazole linkage.