Motilin Receptor

Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。

[Nle13]-Motilin 是一种胃动素 (motilin) 类似物，可作为胃动素受体 motilin receptor 激动剂。

Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.

Idremcinal is a motilin receptor agonist.

Camicinal is a selective motilin receptor agonist (pEC50: 7.9).

MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 is a selective and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 may be useful for gastrointestinal disorders associated with disturbed g

Atilmotin is a gastrointestinal agent for treating motility disorders.

Mitemcinal is a motilin agonist.

RWJ-68022 (Example 9) 是一种环戊烯衍生物，同时也是胃动素受体的拮抗剂。它可以与胃动素和红霉素竞争性结合于胃动素受体位点，并可用于研究胃肠道相关疾病。

Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.

DS-3801b 是一种具有 N-甲基苯胺结构的非大环内酯类 GPR38 激动剂，可用于研究功能性胃肠道疾病。

[Leu13]-Motilin (KW-5139) 为motilin类似物，能够刺激家兔胃肠运动，并在体外以浓度依赖性方式引起胃窦、十二指肠、空肠、回肠以及降结肠的收缩。